[H-3] GBR-12935 BINDING TO THE DOPAMINE TRANSPORTER IS DECREASED IN THE CAUDATE-NUCLEUS IN PARKINSONS-DISEASE

被引:100
作者
JANOWSKY, A
VOCCI, F
BERGER, P
ANGEL, I
ZELNIK, N
KLEINMAN, JE
SKOLNICK, P
PAUL, SM
机构
[1] NIMH,CLIN NEUROSCI BRANCH,MOLEC PHARMACOL SECT,BLDG 10,ROOM 4N214,9000 ROCKVILLE PIKE,BETHESDA,MD 20892
[2] NIMH,NEUROPSYCHIAT BRANCH,CLIN BRAIN STUDIES SECT,BETHESDA,MD 20892
[3] NIADDKD,BIOORGAN CHEM LAB,BETHESDA,MD 20892
[4] NIMH,CLIN NEUROSCI BRANCH,PRECLIN STUDIES SECT,BETHESDA,MD 20892
关键词
D O I
10.1111/j.1471-4159.1987.tb02908.x
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:617 / 621
页数:5
相关论文
共 18 条
[1]  
ALLEN D, 1982, T AM SOC NEUROCHEM, V13, P248
[2]   [H-3] GBR-12935 - A SPECIFIC HIGH-AFFINITY LIGAND FOR LABELING THE DOPAMINE TRANSPORT COMPLEX [J].
BERGER, P ;
JANOWSKY, A ;
VOCCI, F ;
SKOLNICK, P ;
SCHWERI, MM ;
PAUL, SM .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 107 (02) :289-290
[3]   A COMPARISON BETWEEN CENTRIFUGATION AND FILTRATION AS A MEANS TO SEPARATE BOUND AND UNBOUND LIGAND DURING H-3 SPIROPERIDOL BINDING [J].
CSERNANSKY, CA ;
CSERNANSKY, JG ;
HOLLISTER, LE .
JOURNAL OF PHARMACOLOGICAL METHODS, 1985, 13 (03) :187-191
[4]   CHARACTERIZATION OF SODIUM-DEPENDENT [H-3] GBR-12935 BINDING IN BRAIN - A RADIOLIGAND FOR SELECTIVE LABELING OF THE DOPAMINE TRANSPORT COMPLEX [J].
JANOWSKY, A ;
BERGER, P ;
VOCCI, F ;
LABARCA, R ;
SKOLNICK, P ;
PAUL, SM .
JOURNAL OF NEUROCHEMISTRY, 1986, 46 (04) :1272-1276
[5]  
JAVITCH JA, 1984, MOL PHARMACOL, V26, P35
[6]   SODIUM-SENSITIVE COCAINE BINDING TO RAT STRIATAL MEMBRANE - POSSIBLE RELATIONSHIP TO DOPAMINE UPTAKE SITES [J].
KENNEDY, LT ;
HANBAUER, I .
JOURNAL OF NEUROCHEMISTRY, 1983, 41 (01) :172-178
[7]   A PRACTICAL COMPUTER-BASED APPROACH TO THE ANALYSIS OF RADIOLIGAND BINDING EXPERIMENTS [J].
MCPHERSON, GA .
COMPUTER PROGRAMS IN BIOMEDICINE, 1983, 17 (1-2) :107-114
[8]  
PAUL SM, 1981, ARCH GEN PSYCHIAT, V38, P1315
[9]  
PAUL SM, 1984, NEUROBIOLOGY MOOD DI, P846
[10]   DECREASE IN [COCAINE-H-3 BINDING TO THE DOPAMINE TRANSPORTER IN PARKINSONS-DISEASE [J].
PIMOULE, C ;
SCHOEMAKER, H ;
JAVOYAGID, F ;
SCATTON, B ;
AGID, Y ;
LANGER, SZ .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1983, 95 (1-2) :145-146