IMPROVED ASSAYS FOR THE ASSESSMENT OF KAPPA-PROPERTIES AND DELTA-PROPERTIES OF OPIOID LIGANDS

被引：96
作者：
WARD, SJ
PORTOGHESE, PS
TAKEMORI, AE
机构：
[1] UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
[2] UNIV MINNESOTA,COLL PHARM,DEPT MED CHEM,MINNEAPOLIS,MN 55455
来源：
EUROPEAN JOURNAL OF PHARMACOLOGY | 1982年 / 85卷 / 02期
关键词：
D O I：
10.1016/0014-2999(82)90461-7
中图分类号：
R9 [药学];
学科分类号：
1007 ;
摘要：
引用
收藏
页码：163 / 170
页数：8
相关论文
共 27 条
[11]   AGONIST AND ANTAGONIST ACTIONS OF MORPHINE-LIKE DRUGS ON GUINEA-PIG ISOLATED ILEUM [J].
GYANG, EA ;
KOSTERLITZ, HW .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1966, 27 (03) :514-+
[12]   NEW EXAMPLE OF A MORPHINE-SENSITIVE NEURO-EFFECTOR JUNCTION - ADRENERGIC TRANSMISSION IN MOUSE VAS-DEFERENS [J].
HENDERSON, G ;
HUGHES, J ;
KOSTERLITZ, HW .
BRITISH JOURNAL OF PHARMACOLOGY, 1972, 46 (04) :764-766
[13]   EFFECT OF MORPHINE ON ADRENERGIC TRANSMISSION IN MOUSE VAS-DEFERENS ASSESSMENT OF AGONIST AND ANTAGONIST POTENCIES OF NARCOTIC ANALGESICS [J].
HUGHES, J ;
KOSTERLITZ, HW ;
LESLIE, FM .
BRITISH JOURNAL OF PHARMACOLOGY, 1975, 53 (03) :371-381
[14]   ASSESSMENT IN GUINEA-PIG ILEUM AND MOUSE VAS-DEFERENS OF BENZOMORPHANS WHICH HAVE STRONG ANTINOCICEPTIVE ACTIVITY BUT DO NOT SUBSTITUTE FOR MORPHINE IN DEPENDENT MONKEY [J].
HUTCHINSON, M ;
KOSTERLITZ, HW ;
LESLIE, FM ;
WATERFIELD, AA ;
TERENIUS, L .
BRITISH JOURNAL OF PHARMACOLOGY, 1975, 55 (04) :541-546
[15]  
LESLIE FM, 1980, J PHARMACOL EXP THER, V214, P395
[16]   ENDOGENOUS OPIOID PEPTIDES - MULTIPLE AGONISTS AND RECEPTORS [J].
LORD, JAH ;
WATERFIELD, AA ;
HUGHES, J ;
KOSTERLITZ, HW .
NATURE, 1977, 267 (5611) :495-499
[17]  
MARTIN WR, 1978, BR J CLIN PHARM S3, V7, P2735
[18]   SYNTHESIS AND PHARMACOLOGIC CHARACTERIZATION OF AN ALKYLATING ANALOG (CHLORNALTREXAMINE) OF NALTREXONE WITH ULTRA-LONG-LASTING NARCOTIC-ANTAGONIST PROPERTIES [J].
PORTOGHESE, PS ;
LARSON, DL ;
JIANG, JB ;
CARUSO, TP ;
TAKEMORI, AE .
JOURNAL OF MEDICINAL CHEMISTRY, 1979, 22 (02) :168-173
[19]   NOVEL OPIOID RECEPTOR-SITE DIRECTED ALKYLATING AGENT WITH IRREVERSIBLE NARCOTIC ANTAGONISTIC AND REVERSIBLE AGONISTIC ACTIVITIES [J].
PORTOGHESE, PS ;
LARSON, DL ;
SAYRE, LM ;
FRIES, DS ;
TAKEMORI, AE .
JOURNAL OF MEDICINAL CHEMISTRY, 1980, 23 (03) :233-234
[20]   STIMULANT ACTIONS OF VOLATILE ANAESTHETICS ON SMOOTH MUSCLE [J].
RANG, HP .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1964, 22 (02) :356-&
123