AN IMPROVED SYNTHESIS OF 4-FLUOROVERATROLE - EFFICIENT ROUTE TO 6-FLUOROVERATRALDEHYDE AND 6-FLUORO-D,L-DOPA

被引：26

作者：

FURLANO, DC ^{[1
]}

KIRK, KL ^{[1
]}

机构：

[1] NIADDKD,CHEM LAB,BIOCHEM MECHANISMS SECT,BETHESDA,MD 20892

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1986年 / 51卷 / 21期

关键词：

D O I：

10.1021/jo00371a032

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：4073 / 4075

页数：3

共 10 条

[1]

CANTACUZENE D, 1978, SCIENCE WASHINGTON, V204, P1217

[2]

CAREY FA, 1977, ADV ORGANIC CHEM, VB, P275

[3]

CORSE J, 1951, J ORG CHEM, V18, P1345

[4] THE EFFECT OF RING-FLUORINATION ON THE RATE OF O-METHYLATION OF DIHYDROXYPHENYLALANINE (DOPA) BY CATECHOL-O-METHYLTRANSFERASE - SIGNIFICANCE IN THE DEVELOPMENT OF F-18-PETT SCANNING AGENTS [J].

CREVELING, CR ;

KIRK, KL .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1985, 130 (03) :1123-1131

[5] DOPAMINE VISUALIZED IN THE BASAL GANGLIA OF LIVING MAN [J].

GARNETT, ES ;

FIRNAU, G ;

NAHMIAS, C .

NATURE, 1983, 305 (5930) :137-138

[6] UBER ALPHA-HALOGENATHER .13. NEUE VERFAHREN ZUR DARSTELLUNG VON PHENOLALDEHYDEN [J].

GROSS, H ;

RIECHE, A ;

MATTHEY, G .

CHEMISCHE BERICHTE-RECUEIL, 1963, 96 (01) :308-&

[7] SYNTHESIS AND BIOLOGICAL PROPERTIES OF 2-FLUORONOREPINEPHRINES, 5-FLUORONOREPINEPHRINES, AND 6-FLUORONOREPINEPHRINES [J].

KIRK, KL ;

CANTACUZENE, D ;

NIMITKITPAISAN, Y ;

MCCULLOH, D ;

PADGETT, WL ;

DALY, JW ;

CREVELING, CR .

JOURNAL OF MEDICINAL CHEMISTRY, 1979, 22 (12) :1493-1497

[8] THE CHEMISTRY AND BIOLOGY OF RING-FLUORINATED BIOGENIC-AMINES [J].

KIRK, KL ;

CREVELING, CR .

MEDICINAL RESEARCH REVIEWS, 1984, 4 (02) :189-220

[9] IMPROVED SYNTHESIS OF FLUOROVERATROLES AND FLUOROPHENETHYLAMINES VIA ORGANO-LITHIUM REAGENTS [J].

LADD, DL ;

WEINSTOCK, J .

JOURNAL OF ORGANIC CHEMISTRY, 1981, 46 (01) :203-206

[10] The action of acetic acid on 3,4-dimethoxyphenydiazonium borofluoride [J].

Smith, LE ;

Haller, HL .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1934, 56 :237-239

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