NUMBERS OF RECEPTOR-SITES FROM SCATCHARD GRAPHS - FACTS AND FANTASIES

被引:693
作者
KLOTZ, IM
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D O I
10.1126/science.6287580
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O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
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07 ; 0710 ; 09 ;
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页码:1247 / 1249
页数:3
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共 10 条
[1]   ANALYSIS OF MACROMOLECULE-LIGAND BINDING BY DETERMINATION OF STEPWISE EQUILIBRIUM CONSTANTS [J].
FLETCHER, JE ;
SPECTOR, AA ;
ASHBROOK, JD .
BIOCHEMISTRY, 1970, 9 (23) :4580-&
[2]   PROTEIN AFFINITIES FOR SMALL MOLECULES - CONCEPTIONS AND MISCONCEPTIONS [J].
KLOTZ, IM ;
HUNSTON, DL .
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS, 1979, 193 (02) :314-328
[3]  
KLOTZ IM, 1975, J BIOL CHEM, V250, P3001
[4]   THE BINDING OF ORGANIC IONS BY PROTEINS [J].
KLOTZ, IM ;
WALKER, FM ;
PIVAN, RB .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1946, 68 (08) :1486-1490
[5]   THE BINDING OF ORGANIC IONS BY PROTEINS - BUFFER EFFECTS [J].
KLOTZ, IM ;
URQUHART, JM .
JOURNAL OF PHYSICAL AND COLLOID CHEMISTRY, 1949, 53 (01) :100-114
[6]   PROTEIN INTERACTIONS WITH SMALL MOLECULES [J].
KLOTZ, IM .
ACCOUNTS OF CHEMICAL RESEARCH, 1974, 7 (05) :162-168
[7]   LIGAND - A VERSATILE COMPUTERIZED APPROACH FOR CHARACTERIZATION OF LIGAND-BINDING SYSTEMS [J].
MUNSON, PJ ;
RODBARD, D .
ANALYTICAL BIOCHEMISTRY, 1980, 107 (01) :220-239
[8]   DIRECT INVITRO EFFECT OF A SULFONYLUREA TO INCREASE HUMAN FIBROBLAST INSULIN-RECEPTORS [J].
PRINCE, MJ ;
OLEFSKY, JM .
JOURNAL OF CLINICAL INVESTIGATION, 1980, 66 (03) :608-611
[9]   PENTOBARBITAL - DUAL ACTIONS TO INCREASE BRAIN BENZODIAZEPINE RECEPTOR AFFINITY [J].
SKOLNICK, P ;
MONCADA, V ;
BARKER, JL ;
PAUL, SM .
SCIENCE, 1981, 211 (4489) :1448-1450
[10]  
SUTER P, 1976, J BIOL CHEM, V251, P5986