RESOLUTION OF 5,6-DIHYDROXY-2-(N,N-DI-NORMAL-PROPYLAMINO)TETRALIN IN RELATION TO THE STRUCTURAL AND STEREOCHEMICAL REQUIREMENTS FOR CENTRALLY ACTING DOPAMINE AGONISTS

被引：23
作者：
GROL, CJ
JANSEN, LJ
ROLLEMA, H
机构：
来源：
JOURNAL OF MEDICINAL CHEMISTRY | 1985年 / 28卷 / 05期
关键词：
D O I：
10.1021/jm50001a024
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
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页码：679 / 683
页数：5
相关论文
共 21 条
[1]   BICYCLIC AND TRICYCLIC ERGOLINE PARTIAL STRUCTURES - RIGID 3-(2-AMINOETHYL)PYRROLES AND 3-(2-AMINOETHYL)PYRAZOLE AND 4-(2-AMINOETHYL)PYRAZOLE AS DOPAMINE AGONISTS [J].
BACH, NJ ;
KORNFELD, EC ;
JONES, ND ;
CHANEY, MO ;
DORMAN, DE ;
PASCHAL, JW ;
CLEMENS, JA ;
SMALSTIG, EB .
JOURNAL OF MEDICINAL CHEMISTRY, 1980, 23 (05) :481-491
[2]   DOPAMINE-RECEPTORS IN RAT-BRAIN REGIONS - OPTIMAL CONDITIONS FOR H-3-AGONIST BINDING, PH DEPENDENCY AND LACK OF INHIBITION BY ASCORBIC-ACID [J].
BACOPOULOS, NG .
BIOCHEMICAL PHARMACOLOGY, 1982, 31 (19) :3085-3091
[3]   PROPOSED DOPAMINERGIC PHARMACOPHORE OF LERGOTRILE, PERGOLIDE, AND RELATED ERGOT ALKALOID DERIVATIVES [J].
CANNON, JG ;
DEMOPOULOS, BJ ;
LONG, JP ;
FLYNN, JR ;
SHARABI, FM .
JOURNAL OF MEDICINAL CHEMISTRY, 1981, 24 (03) :238-240
[4]   DIFFERENTIATION OF DOPAMINE MECHANISMS MEDIATING STEREOTYPED BEHAVIOR AND HYPERACTIVITY IN NUCLEUS ACCUMBENS AND CAUDATE-PUTAMEN [J].
COSTALL, B ;
NAYLOR, RJ ;
CANNON, JG ;
LEE, T .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1977, 29 (06) :337-342
[5]   SYNTHESIS, RESOLUTION, ABSOLUTE STEREOCHEMISTRY, AND ENANTIOSELECTIVITY OF 3',4'-DIHYDROXYNOMIFENSINE [J].
DANDRIDGE, PA ;
KAISER, C ;
BRENNER, M ;
GAITANOPOULOS, D ;
DAVIS, LD ;
WEBB, RL ;
FOLEY, JJ ;
SARAU, HM .
JOURNAL OF MEDICINAL CHEMISTRY, 1984, 27 (01) :28-35
[6]   EFFECT OF DIHYDROXY-2-AMINOTETRALIN DERIVATIVES ON DOPAMINE METABOLISM IN THE RAT STRIATUM [J].
FEENSTRA, MGP ;
ROLLEMA, H ;
HORN, AS ;
DIJKSTRA, D ;
GROL, CJ ;
WESTERINK, BHC ;
WESTERBRINK, A .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1980, 310 (03) :219-225
[7]  
FREEMAN HS, 1981, 1ST P MED CHEM S CAM
[8]  
GROL CJ, 1983, J PHARM PHARM, V29, P153
[9]   MONOPHENOLIC 2-(DIPROPYLAMINO)INDANS AND RELATED-COMPOUNDS - CENTRAL DOPAMINE-RECEPTOR STIMULATING ACTIVITY [J].
HACKSELL, U ;
ARVIDSSON, LE ;
SVENSSON, U ;
NILSSON, JLG ;
WIKSTROM, H ;
LINDBERG, P ;
SANCHEZ, D ;
HJORTH, S ;
CARLSSON, A ;
PAALZOW, L .
JOURNAL OF MEDICINAL CHEMISTRY, 1981, 24 (04) :429-434
[10]   FACILE SYNTHESES OF POTENT DOPAMINERGIC AGONISTS AND THEIR EFFECTS ON NEUROTRANSMITTER RELEASE [J].
HORN, AS ;
GROL, CJ ;
DIJKSTRA, D ;
MULDER, AH .
JOURNAL OF MEDICINAL CHEMISTRY, 1978, 21 (08) :825-828
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