HIGHLY SELECTIVE AND SPECIFIC ANTAGONISM OF CENTRAL AND PERIPHERAL ALPHA-2-ADRENOCEPTORS BY ATIPAMEZOLE

被引:1
|
作者
VIRTANEN, R
SAVOLA, JM
SAANO, V
机构
[1] UNIV OULU,DEPT PHARMACOL,SF-90100 OULU 10,FINLAND
[2] UNIV KUOPIO,DEPT PHARMACOL & TOXICOL,KUOPIO,FINLAND
来源
ARCHIVES INTERNATIONALES DE PHARMACODYNAMIE ET DE THERAPIE | 1989年 / 297卷
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:190 / 204
页数:15
相关论文
共 50 条
  • [1] ALPHA-2-ADRENOCEPTORS AND VIGILANCE IN CATS - ANTAGONISM OF MEDETOMIDINE SEDATION BY ATIPAMEZOLE
    STENBERG, D
    PORKKAHEISKANEN, T
    TOPPILA, J
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1993, 238 (2-3) : 241 - 247
  • [2] CENTRAL ALPHA-2-ADRENOCEPTORS REGULATE CENTRAL AND PERIPHERAL FUNCTIONS
    FORNAI, F
    BLANDIZZI, C
    DELTACCA, M
    PHARMACOLOGICAL RESEARCH, 1990, 22 (05) : 541 - 554
  • [3] CHARACTERIZATION OF [H-3] ATIPAMEZOLE AS A RADIOLIGAND FOR ALPHA-2-ADRENOCEPTORS
    SJOHOLM, B
    VOUTILAINEN, R
    LUOMALA, K
    SAVOLA, JM
    SCHEININ, M
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1992, 215 (01) : 109 - 117
  • [4] CENTRAL ALPHA-2-ADRENOCEPTORS ARE HIGHLY STEREOSELECTIVE FOR DEXMEDETOMIDINE, THE DEXTRO ENANTIOMER OF MEDETOMIDINE
    SAVOLA, JM
    VIRTANEN, R
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1991, 195 (02) : 193 - 199
  • [5] INVITRO DETERMINATION OF THE RELATIVE SELECTIVITY OF IFENPRODIL FOR BLOCKING PERIPHERAL AND CENTRAL ALPHA-1-ADRENOCEPTORS AND ALPHA-2-ADRENOCEPTORS
    CASADAMONT, M
    CATHALA, F
    LANGER, SZ
    MASSINGHAM, R
    MORET, C
    BRITISH JOURNAL OF PHARMACOLOGY, 1981, 74 (01) : P257 - P258
  • [6] A ROLE FOR CENTRAL POSTSYNAPTIC ALPHA-2-ADRENOCEPTORS IN GLUCOREGULATION
    SMYTHE, GA
    EDWARDS, SR
    BRAIN RESEARCH, 1991, 562 (02) : 225 - 229
  • [7] STUDIES ON RX781094 - A SELECTIVE, POTENT AND SPECIFIC ANTAGONIST OF ALPHA-2-ADRENOCEPTORS
    DOXEY, JC
    ROACH, AG
    SMITH, CFC
    BRITISH JOURNAL OF PHARMACOLOGY, 1983, 78 (03) : 489 - 505
  • [8] ACTIONS OF TIZANIDINE ON ALPHA-1-ADRENOCEPTORS AND ALPHA-2-ADRENOCEPTORS IN THE PERIPHERAL-TISSUES
    TAKAYANAGI, I
    KONNO, F
    ISHII, C
    TAKEMASA, T
    YANAGIDA, Y
    SHIMIZU, M
    MORI, H
    SUGANE, H
    GENERAL PHARMACOLOGY-THE VASCULAR SYSTEM, 1984, 15 (03): : 239 - 241
  • [9] ACUTE AND CHRONIC EFFECTS OF RESERPINE ON BIOCHEMICAL AND FUNCTIONAL PARAMETERS OF CENTRAL AND PERIPHERAL ALPHA-2-ADRENOCEPTORS
    UGEDO, L
    GARRO, MA
    PINEDA, J
    GIRALT, MT
    MIRALLES, A
    OLMOS, G
    GARCIASEVILLA, JA
    MENARGUES, A
    OBACH, R
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1993, 239 (1-3) : 149 - 157
  • [10] FUNCTIONAL EVIDENCE FOR HETEROGENEITY OF PERIPHERAL PREJUNCTIONAL ALPHA-2-ADRENOCEPTORS
    CONNAUGHTON, S
    DOCHERTY, JR
    BRITISH JOURNAL OF PHARMACOLOGY, 1990, 101 (02) : 285 - 290