THE DESIGN OF FULL AGONISTS FOR THE CORTICAL MUSCARINIC RECEPTOR

被引:0
|
作者
SAUNDERS, J [1 ]
FREEDMAN, SB [1 ]
机构
[1] MERCK SHARP & DOHME LTD,RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:70 / 75
页数:6
相关论文
共 50 条
  • [21] Differential Rho-kinase dependency of full and partial muscarinic receptor agonists in airway smooth muscle contraction
    Schaafsma, D
    Boterman, M
    de Jong, AM
    Hovens, I
    Penninks, JM
    Nelemans, SA
    Meurs, H
    Zaagsma, J
    BRITISH JOURNAL OF PHARMACOLOGY, 2006, 147 (07) : 737 - 743
  • [22] THE RATIONAL DESIGN AND SYNTHESIS OF HAPTENS HAVING SPECIFIC ACTIVITY AS FULL AGONISTS OR FULL ANTAGONISTS AT THE BENZODIAZEPINE RECEPTOR
    FRYER, RI
    GU, ZQ
    LIFE SCIENCES, 1990, 47 (10) : 833 - 840
  • [24] A NOVEL SERIES OF NONQUATERNARY OXADIAZOLES ACTING AS FULL AGONISTS AT MUSCARINIC RECEPTORS
    FREEDMAN, SB
    HARLEY, EA
    PATEL, S
    NEWBERRY, NR
    GILBERT, MJ
    MCKNIGHT, AT
    TANG, JK
    MAGUIRE, JJ
    MUDUNKOTUWA, NT
    BAKER, R
    STREET, LJ
    MACLEOD, AM
    SAUNDERS, J
    IVERSEN, LL
    BRITISH JOURNAL OF PHARMACOLOGY, 1990, 101 (03) : 575 - 580
  • [25] THE DESIGN AND PHARMACOLOGY OF NOVEL SELECTIVE MUSCARINIC AGONISTS AND ANTAGONISTS
    LAMBRECHT, G
    GROSS, J
    HACKSELL, U
    HERMANNI, U
    HILDEBRANDT, C
    HOU, X
    MOSER, U
    NILSSON, BM
    PFAFF, O
    WAELBROECK, M
    WEHRLE, J
    MUTSCHLER, E
    LIFE SCIENCES, 1995, 56 (11-12) : 815 - 822
  • [26] RECENT ADVANCES IN THE DESIGN AND CHARACTERIZATION OF MUSCARINIC AGONISTS AND ANTAGONISTS
    JAEN, JC
    DAVIS, RE
    ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 29, 1994, 29 : 23 - 32
  • [27] Muscarinic receptor agonists and antagonists in the treatment of Alzheimer's Disease
    Clader, JW
    Wang, YG
    CURRENT PHARMACEUTICAL DESIGN, 2005, 11 (26) : 3353 - 3361
  • [28] Synthesis and pharmacological evaluation of dimeric muscarinic acetylcholine receptor agonists
    Christopoulos, A
    Grant, MKO
    Ayoubzadeh, N
    Kim, ON
    Sauerberg, P
    Jeppesen, L
    El-Fakahany, EE
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2001, 298 (03) : 1260 - 1268
  • [29] CHANGES IN VAGAL ACTIVITY AND RESPONSE TO MUSCARINIC RECEPTOR AGONISTS WITH AGE
    KELLIHER, GJ
    CONAHAN, ST
    JOURNALS OF GERONTOLOGY, 1980, 35 (06): : 842 - 849
  • [30] MUSCARINIC-M(1) RECEPTOR AGONIST ACTIONS OF MUSCARINIC RECEPTOR AGONISTS IN RABBIT VAS-DEFERENS
    SHANNON, HE
    SAWYER, BD
    BEMIS, KG
    BYMASTER, FP
    HEATH, I
    MITCH, CH
    WARD, JS
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1993, 232 (01) : 47 - 57