5-CINNAMOYL-6-AMINOURACIL DERIVATIVES AS NOVEL ANTICANCER AGENTS - SYNTHESIS, BIOLOGICAL EVALUATION, AND STRUCTURE ACTIVITY RELATIONSHIPS

被引：31
作者：
BERNIER, JL
HENICHART, JP
WARIN, V
TRENTESAUX, C
JARDILLIER, JC
机构：
[1] UNIV LILLE 1,CNRS,ERA 465,F-59655 VILLENEUVE DASCQ,FRANCE
[2] FAC PHARM REIMS,BIOCHIM LAB,F-51100 REIMS,FRANCE
来源：
JOURNAL OF MEDICINAL CHEMISTRY | 1985年 / 28卷 / 04期
关键词：
D O I：
10.1021/jm00382a020
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
引用
收藏
页码：497 / 502
页数：6
相关论文
共 19 条
[1]  
BERLINGER LJ, 1976, SPIN LABELLING THEOR, V1
[2]  
BERLINGER LJ, 1979, SPIN LABELLING THEOR, V2
[3]  
Bernier J. L., 1976, B SOC CHIM FR, V3, P617
[4]   ELECTRON-SPIN-RESONANCE STUDY OF INTERCALATION - QUANTITATIVE-EVALUATION OF DRUG-DNA BINDING THROUGH COMPETITION WITH A SPIN-LABELED 9-AMINOACRIDINE [J].
BERNIER, JL ;
HENICHART, JP ;
CATTEAU, JP .
ANALYTICAL BIOCHEMISTRY, 1981, 117 (01) :12-17
[5]  
BERNIER JL, 1977, EUR J MED CHEM, V12, P341
[6]  
BERNIER JL, 1980, J PHARM SCI, V69, P1343, DOI 10.1002/jps.2600691128
[7]  
BERNIER JL, 1977, EUR J MED CHEM, V12, P239
[8]   REACTIONS OF 1,3-DIMETHYL-5,6-DIAMINOURACIL [J].
BLICKE, FF ;
GODT, HC .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1954, 76 (10) :2798-2800
[9]   POTENTIAL ANTITUMOR AGENTS 16.4'-(ACRIDIN-9-YLAMINO)METHANESULFONANILIDES [J].
CAIN, BF ;
ATWELL, GJ ;
DENNY, WA .
JOURNAL OF MEDICINAL CHEMISTRY, 1975, 18 (11) :1110-1117
[10]   EXPERIMENTAL ANTITUMOR PROPERTIES OF 3 CONGENERS OF ACRIDYLMETHANESULFONANILIDE (AMSA) SERIES [J].
CAIN, BF ;
ATWELL, GJ .
EUROPEAN JOURNAL OF CANCER, 1974, 10 (08) :539-549
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