DIOXIDES OF BICYCLIC THIADIAZINES - A NEW FAMILY OF SMOOTH-MUSCLE RELAXANTS

被引:16
作者
CASTRO, A
MARTINEZ, A
CARDELUS, I
LLENAS, J
机构
[1] CSIC, INST QUIM MED, E-28006 MADRID, Spain
[2] LAB ALMIRALL SA, E-08024 BARCELONA, Spain
关键词
D O I
10.1016/0968-0896(95)00012-6
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
The synthesis of dioxides of bicyclic thiadiazine related to diazoxide has been achieved. In a preliminary test, some of these compounds show smooth muscle relaxation similar to that obtained with the reference standard diazoxide.
引用
收藏
页码:179 / 185
页数:7
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