PESTICIDAL ACTIVITIES OF SOME 3-ARYL-4-METHYLPYRAZOLO[3,4-B][1,5]BENZODIAZEPINES AND 4-ARYL-2-IMINO-5-METHYL-1,3-THIAZINO[4,5-B][1,5]BENZODIAZEPINES

被引：21
作者：
KHAN, MH
BANO, Q
NIZAMUDDIN
机构：
[1] Agrochemical Research Laboratory, Department of Chemistry, University of Gorakhpur
来源：
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY | 1995年 / 43卷 / 10期
关键词：
PYRAZOLO[3,4-B][1,5]BENZODIAZEPINES; THIAZINO[4,5-B][1,5]BENZODIAZEPINES; INSECTICIDAL AND FUNGISTATIC ACTIVITIES;
D O I：
10.1021/jf00058a032
中图分类号：
S [农业科学];
学科分类号：
09 ;
摘要：
A number of 3-aryl-4-methylpyrazolo[3,4-b][1,5]benzodiazepines and 4-aryl-2-imino-5-methyl-1,3-thiazino[4,5-b][1,5]benzodiazepines have been synthesized from 3-(arylmethylene)-4-methyl-1,5-benzodiazepin-2-one by cyclocondensation with hydrazine hydrate and thiourea in basic medium, respectively. All of the compounds were evaluated for their insecticidal and fungistatic activities, and the results are compared with the standard insecticide Propoxure and the standard fungicide Maneb. Some structure-activity relationships are discussed on the basis of screening data.
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页码：2719 / 2721
页数：3
相关论文
共 12 条
  • [1] ALHADEFF M, 1977, MED ACTUAL, V13, P521
  • [2] ATWAL K, 1987, Patent No. 4650797
  • [3] CANJOLLE R, 1989, EUR J MED CHEM, V24, P287
  • [4] CLIFFORD DP, 1976, PESTIC SCI, V7, P453, DOI 10.1002/ps.2780070506
  • [5] FENG J, 1984, YIYAO GANGYE, V2, P12
  • [6] HOLLOWOOD J, 1986, Patent No. 189972
  • [7] KHAN M H, 1992, Indian Journal of Pharmaceutical Sciences, V54, P128
  • [8] KULKARNI SU, 1976, J INDIAN CHEM SOC, V53, P279
  • [9] MENDELSON WB, 1982, PHARM BENZODIAZEPINE, P375
  • [10] ROMA G, 1983, FARMACO-ED SCI, V38, P546
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