KETOCONAZOLE BINDS TO GLUCOCORTICOID RECEPTORS AND EXHIBITS GLUCOCORTICOID ANTAGONIST ACTIVITY IN CULTURED-CELLS

被引：113

作者：

LOOSE, DS ^{[1
]}

STOVER, EP ^{[1
]}

FELDMAN, D ^{[1
]}

机构：

[1] STANFORD UNIV,MED CTR,SCH MED,DEPT MED,STANFORD,CA 94305

来源：

JOURNAL OF CLINICAL INVESTIGATION | 1983年 / 72卷 / 01期

关键词：

D O I：

10.1172/JCI110982

中图分类号：

R-3 [医学研究方法]; R3 [基础医学];

学科分类号：

1001 ;

摘要：

引用

页码：404 / 408

页数：5

共 15 条

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[9] MOLECULAR MODIFICATIONS OF ANTI-ALDOSTERONE COMPOUNDS - EFFECTS ON AFFINITY OF SPIRONOLACTONES FOR RENAL ALDOSTERONE RECEPTORS [J].

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[10] KETOCONAZOLE BLOCKS ADRENAL STEROIDOGENESIS BY INHIBITING CYTOCHROME-P450-DEPENDENT ENZYMES [J].

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