CYP3A5 EXPRESSION IN HUMAN ENTEROCYTES

被引:0
作者
JANARDAN, SK [1 ]
LOWN, KS [1 ]
GHOSH, M [1 ]
KOLARS, JC [1 ]
WATKINS, PB [1 ]
机构
[1] UNIV MICHIGAN,DEPT MED,ANN ARBOR,MI 48109
关键词
D O I
暂无
中图分类号
R57 [消化系及腹部疾病];
学科分类号
摘要
引用
收藏
页码:A241 / A241
页数:1
相关论文
共 50 条
[11]   In vitro metabolism of cyclosporine A by human kidney CYP3A5 [J].
Dai, Y ;
Iwanaga, K ;
Lin, YS ;
Hebert, MF ;
Davis, CL ;
Huang, WL ;
Kharasch, ED ;
Thummel, KE .
BIOCHEMICAL PHARMACOLOGY, 2004, 68 (09) :1889-1902
[12]   CYP3A5 phenotyping of human liver microsomes with vincristine [J].
Dennison, Jennifer B. ;
Jones, David R. ;
Renbarger, Jamie L. ;
Hall, Stephen D. .
DRUG METABOLISM REVIEWS, 2006, 38 :210-210
[13]   In vitro and in vivo analysis of the human cyp3a5 promoter [J].
Nem, D. ;
Qiu, H. ;
Nestler, S. ;
Goedtel-Armbrust, U. ;
Wojnowski, L. .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 2010, 381 :88-88
[14]   Association of the CYP3A5 A6986G (CYP3A5*3) polymorphism with saquinavir pharmacokinetics [J].
Fröhlich, M ;
Hoffmann, MM ;
Burhenne, J ;
Mikus, G ;
Weiss, J ;
Haefeli, WE .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 2004, 58 (04) :443-444
[15]   PharmVar GeneFocus: CYP3A5 [J].
Rodriguez-Antona, Cristina ;
Savieo, Jessica L. ;
Lauschke, Volker M. ;
Sangkuhl, Katrin ;
Drogemoller, Britt, I ;
Wang, Danxin ;
Schaik, Ron N. H. ;
Gilep, Andrei A. ;
Peter, Arul P. ;
Boone, Erin C. ;
Ramey, Bronwyn E. ;
Klein, Teri E. ;
Whirl-Carrillo, Michelle ;
Pratt, Victoria M. ;
Gaedigk, Andrea .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 2022, 112 (06) :1159-1171
[16]   Comparative analysis of CYP3A expression in human liver suggests only a minor role for CYP3A5 in drug metabolism [J].
Westlind-Johnsson, A ;
Malmebo, S ;
Johansson, A ;
Otter, C ;
Andersson, TB ;
Johansson, I ;
Edwards, RJ ;
Boobis, AR ;
Ingelman-Sundberg, M .
DRUG METABOLISM AND DISPOSITION, 2003, 31 (06) :755-761
[17]   Differential drug-induced mRNA expression of human CYP3A4 compared to CYP3A5, CYP3A7 and CYP3A43 [J].
Krusekopf, S ;
Roots, I ;
Kleeberg, U .
EUROPEAN JOURNAL OF PHARMACOLOGY, 2003, 466 (1-2) :7-12
[18]   In vitro metabolism of cyclosporine A by human kidney microsomal CYP3A5 [J].
Dai, Y ;
Iwanaga, K ;
Lin, YS ;
Huang, W ;
Thummel, KE .
DRUG METABOLISM REVIEWS, 2003, 35 :188-188
[19]   Variability in Expression of CYP3A5 in Human Fetal Liver (vol 43, pg 1286, 2015) [J].
Vyhlidal, C. A. ;
Pearce, R. E. ;
Gaedigk, R. ;
Calamia, J. C. ;
Shuster, D. L. ;
Thummel, K. E. ;
Leeder, J. S. .
DRUG METABOLISM AND DISPOSITION, 2016, 44 (09) :1459-1459
[20]   Apparent high CYP3A5 expression is required for significant metabolism of vincristine by human cryopreserved hepatocytes [J].
Dennison, Jennifer B. ;
Mohutsky, Michael A. ;
Barbuch, Robert J. ;
Wrighton, Steven A. ;
Hall, Stephen D. .
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2008, 327 (01) :248-257