DISTRIBUTION OF MUSCARINIC RECEPTOR SUBTYPES IN RAT-BRAIN AS DETERMINED IN BINDING-STUDIES WITH AF-DX 116 AND PIRENZEPINE

被引:135
作者
GIRALDO, E [1 ]
HAMMER, R [1 ]
LADINSKY, H [1 ]
机构
[1] BOEHRINGER INGELHEIM ZENT GMBH,FL BIOCHEM,D-6507 INGELHEIM,FED REP GER
关键词
D O I
10.1016/0024-3205(87)90031-2
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:833 / 840
页数:8
相关论文
共 19 条
[1]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[2]  
ENGEL W, FED P
[3]   CARDIOSELECTIVE PROFILE OF AF-DX-116, A MUSCARINE M2 RECEPTOR ANTAGONIST [J].
GIACHETTI, A ;
MICHELETTI, R ;
MONTAGNA, E .
LIFE SCIENCES, 1986, 38 (18) :1663-1672
[4]   MUSCARINIC RECEPTOR SUBTYPES - M1 AND M2 BIOCHEMICAL AND FUNCTIONAL-CHARACTERIZATION [J].
HAMMER, R ;
GIACHETTI, A .
LIFE SCIENCES, 1982, 31 (26) :2991-2998
[5]   BINDING PROFILE OF A NOVEL CARDIOSELECTIVE MUSCARINE RECEPTOR ANTAGONIST, AF-DX 116, TO MEMBRANES OF PERIPHERAL-TISSUES AND BRAIN IN THE RAT [J].
HAMMER, R ;
GIRALDO, E ;
SCHIAVI, GB ;
MONFERINI, E ;
LADINSKY, H .
LIFE SCIENCES, 1986, 38 (18) :1653-1662
[6]   PIRENZEPINE DISTINGUISHES BETWEEN DIFFERENT SUBCLASSES OF MUSCARINIC RECEPTORS [J].
HAMMER, R ;
BERRIE, CP ;
BIRDSALL, NJM ;
BURGEN, ASV ;
HULME, EC .
NATURE, 1980, 283 (5742) :90-92
[7]  
HAMMER R, 1986, TRENDS PHARMSCI S, V2, P33
[8]  
HEINZEL G, 1982, PHARMACOKINETICS DRU, P207
[9]  
HIRSCHOWITZ BI, 1984, TRENDS PHARM SCI S
[10]  
IVERSEN LL, 1986, TRENDS PHARMACOL SCI, P44