BENZODIAZEPINE RECEPTORS - MODE OF INTERACTION OF AGONISTS AND ANTAGONISTS

被引:0
作者
MOHLER, H [1 ]
机构
[1] F HOFFMANN LA ROCHE & CO LTD,PHARMACEUT RES DEPT,CH-4002 BASEL,SWITZERLAND
关键词
D O I
暂无
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:247 / 254
页数:8
相关论文
共 41 条
[1]   INVITRO AND INVIVO INHIBITION BY ZOPICLONE OF BENZODIAZEPINE BINDING TO RODENT BRAIN RECEPTORS [J].
BLANCHARD, JC ;
BOIREAU, A ;
GARRET, C ;
JULOU, L .
LIFE SCIENCES, 1979, 24 (26) :2417-2420
[2]   BENZODIAZEPINE ANTAGONIST RO 15-1788 - NEUROLOGICAL AND BEHAVIORAL-EFFECTS [J].
BONETTI, EP ;
PIERI, L ;
CUMIN, R ;
SCHAFFNER, R ;
PIERI, M ;
GAMZU, ER ;
MULLER, RKM ;
HAEFELY, W .
PSYCHOPHARMACOLOGY, 1982, 78 (01) :8-18
[3]   INTERACTION OF CONVULSIVE LIGANDS WITH BENZODIAZEPINE RECEPTORS [J].
BRAESTRUP, C ;
SCHMIECHEN, R ;
NEEF, G ;
NIELSEN, M ;
PETERSEN, EN .
SCIENCE, 1982, 216 (4551) :1241-1243
[4]   URINARY AND BRAIN BETA-CARBOLINE-3-CARBOXYLATES AS POTENT INHIBITORS OF BRAIN BENZODIAZEPINE RECEPTORS [J].
BRAESTRUP, C ;
NIELSEN, M ;
OLSEN, CE .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (04) :2288-2292
[5]   GABA REDUCES BINDING OF H-3-LABELED METHYL BETA-CARBOLINE-3-CARBOXYLATE TO BRAIN BENZODIAZEPINE RECEPTORS [J].
BRAESTRUP, C ;
NIELSEN, M .
NATURE, 1981, 294 (5840) :472-474
[6]  
BRAESTRUP C, 1981, J NEUROCHEM, V37, P334
[7]   ETHYL BETA-CARBOLINE CARBOXYLATE LOWERS SEIZURE THRESHOLD AND ANTAGONIZES FLURAZEPAM-INDUCED SEDATION IN RATS [J].
COWEN, PJ ;
GREEN, AR ;
NUTT, DJ ;
MARTIN, IL .
NATURE, 1981, 290 (5801) :54-55
[8]  
DARRAGH A, 1981, LANCET, V2, P8
[9]  
DECARVALHO LP, 1983, NATURE
[10]   ETHYL BETA-CARBOLINE-3-CARBOXYLATE REVERSES THE DIAZEPAM EFFECT ON CEREBELLAR CYCLIC-GMP [J].
FUJIMOTO, M ;
KAWASAKI, K ;
MATSUSHITA, A ;
OKABAYASHI, T .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 80 (2-3) :259-262