SRN1 REACTIONS IN IMIDAZO[1,2-A]PYRIDINE SERIES

被引：40
作者：
VANELLE, P
MALDONADO, J
MADADI, N
GUEIFFIER, A
TEULADE, JC
CHAPAT, JP
CROZET, MP
机构：
[1] FAC PHARM MONTPELLIER,CNRS,CHIM ORGAN PHARMACEUT LAB,F-34006 MONTPELLIER,FRANCE
[2] UNIV DROIT ECON & SCI AIX MARSEILLE,FAC SCI & TECH ST JEROME,CNRS,F-13397 MARSEILLE 13,FRANCE
来源：
TETRAHEDRON LETTERS | 1990年 / 31卷 / 21期
关键词：
D O I：
10.1016/S0040-4039(00)89012-7
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
2-Chloromethyl-3-nitroimidazo[1,2-a]pyridine is shown for the first time to react with 2-nitropropane salts by an SRN1 mechanism to give excellent yield of isopropylidene derivative formed from the C-alkylation product by loss of nitrous acid. © 1990.
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页码：3013 / 3016
页数：4
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