OPIATE BINDING IN THE RAT SPINAL-CORD - EVIDENCE FOR MU AND DELTA SITES

被引:20
作者
TRAYNOR, JR [1 ]
RANCE, MJ [1 ]
机构
[1] ICI LTD,DIV PHARMACEUT,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
关键词
D O I
10.1016/0143-4179(84)90032-5
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:81 / 84
页数:4
相关论文
共 9 条
[1]   SPECTRUM OF THE MU-BINDING, DELTA-BINDING AND KAPPA-BINDING SITES IN HOMOGENATES OF RAT-BRAIN [J].
GILLAN, MGC ;
KOSTERLITZ, HW .
BRITISH JOURNAL OF PHARMACOLOGY, 1982, 77 (03) :461-468
[2]   INTERACTION OF SELECTIVE MU-LIGANDS AND DELTA-LIGANDS WITH THE KAPPA-2 SUBTYPE OF OPIATE BINDING-SITES [J].
GOUARDERES, C ;
ATTALI, B ;
AUDIGIER, Y ;
CROS, J .
LIFE SCIENCES, 1983, 33 :175-178
[3]  
GOUARDERES C, 1981, ADV ENDOGENOUS EXOGE, P18
[4]  
HYLDEN J L K, 1983, European Journal of Pharmacology, V86, P95
[5]  
MARTIN WR, 1976, J PHARMACOL EXP THER, V197, P517
[6]   MULTIPLE OPIATE BINDING-SITES IN RAT SPINAL-CORD [J].
TRAYNOR, JR ;
KELLY, PD ;
RANCE, MJ .
LIFE SCIENCES, 1982, 31 (12-1) :1377-1380
[7]   INVIVO EVIDENCE FOR MULTIPLE OPIATE RECEPTORS MEDIATING ANALGESIA IN THE RAT SPINAL-CORD [J].
TUNG, AS ;
YAKSH, TL .
BRAIN RESEARCH, 1982, 247 (01) :75-83
[8]   SPINAL ANALGESIA - COMPARISON OF THE MU AGONIST MORPHINE AND THE KAPPA AGONIST ETHYLKETAZOCINE [J].
WOOD, PL ;
RACKHAM, A ;
RICHARD, J .
LIFE SCIENCES, 1981, 28 (19) :2119-2125
[9]   SPINAL OPIATE ANALGESIA - CHARACTERISTICS AND PRINCIPLES OF ACTION [J].
YAKSH, TL .
PAIN, 1981, 11 (03) :293-346