A MILD AND EFFICIENT METHOD FOR THE PREPARATION OF GUANIDINES

被引：149

作者：

POSS, MA

IWANOWICZ, E

REID, JA

LIN, J

GU, ZX

机构：

来源：

TETRAHEDRON LETTERS | 1992年 / 33卷 / 40期

关键词：

ACYLGUANIDINE; ACYLTHIOUREA; GUANIDINE; WATER SOLUBLE CARBODIIMIDE;

D O I：

10.1016/S0040-4039(00)61092-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A mild and efficient method for the preparation of guanidines by reaction of an acylated thiourea with an amine followed by removal of the acyl group(s) from the intermediate acylguanidine is reported.

引用

页码：5933 / 5936

页数：4

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