MECHANISM OF ACTION AND SYSTEMIC AND REGIONAL HEMODYNAMICS OF THE POTASSIUM CHANNEL ACTIVATOR BRL34915 AND ITS ENANTIOMERS

被引:129
作者
HOF, RP
QUAST, U
COOK, NS
BLARER, S
机构
关键词
D O I
10.1161/01.RES.62.4.679
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:679 / 686
页数:8
相关论文
共 38 条
[1]   SYNTHESIS AND ANTIHYPERTENSIVE ACTIVITY OF 4-(CYCLIC AMIDO)-2H-1-BENZOPYRANS [J].
ASHWOOD, VA ;
BUCKINGHAM, RE ;
CASSIDY, F ;
EVANS, JM ;
FARUK, EA ;
HAMILTON, TC ;
NASH, DJ ;
STEMP, G ;
WILLCOCKS, K .
JOURNAL OF MEDICINAL CHEMISTRY, 1986, 29 (11) :2194-2201
[2]   ACTIONS OF VARIOUS MUSCARINIC AGONISTS ON MEMBRANE-POTENTIAL, POTASSIUM EFFLUX, AND CONTRACTION OF LONGITUDINAL MUSCLE OF GUINEA-PIG INTESTINE [J].
BOLTON, TB ;
CLARK, JP .
BRITISH JOURNAL OF PHARMACOLOGY, 1981, 72 (02) :319-334
[3]   EVIDENCE THAT THE MECHANISM OF THE INHIBITORY-ACTION OF PINACIDIL IN RAT AND GUINEA-PIG SMOOTH-MUSCLE DIFFERS FROM THAT OF GLYCERYL TRINITRATE [J].
BRAY, KM ;
NEWGREEN, DT ;
SMALL, RC ;
SOUTHERTON, JS ;
TAYLOR, SG ;
WEIR, SW ;
WESTON, AH .
BRITISH JOURNAL OF PHARMACOLOGY, 1987, 91 (02) :421-429
[4]  
BUCKINGHAM R E, 1986, British Journal of Pharmacology, V87, p78P
[5]  
BUCKINGHAM RE, 1986, J CARDIOVASC PHARM, V8, P798
[6]   MECHANISMS OF CALCIUM ANTAGONIST-INDUCED VASODILATION [J].
CAUVIN, C ;
LOUTZENHISER, R ;
VANBREEMEN, C .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1983, 23 :373-396
[8]  
COOK NS, 1987, IN PRESS J CARDIOVAS
[9]   RELATIVE CONTRIBUTIONS OF CA2+INFLUX AND CELLULAR CA2+RELEASE DURING DRUG-INDUCED ACTIVATION OF RABBIT AORTA [J].
DETH, R ;
VANBREEM, C .
PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY, 1974, 348 (01) :13-22
[10]  
DRAPER NR, 1981, APPLIED REGRESSION A, P85