THE 5-HYDROXYTRYPTAMINE 5-HT1D RECEPTOR SUBTYPE IS NEGATIVELY COUPLED TO ADENYLATE-CYCLASE IN CALF SUBSTANTIA NIGRA

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作者
SCHOEFFTER, P [1 ]
WAEBER, C [1 ]
PALACIOS, JM [1 ]
HOYER, D [1 ]
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[1] SANDOZ LTD,PRECLIN RES,BLDG 386-525,CH-4002 BASEL,SWITZERLAND
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R9 [药学];
学科分类号
1007 ;
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页码:602 / 608
页数:7
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[41]   5-HT (SEROTONIN) STIMULATED ADENYLATE-CYCLASE ACTIVITY IS MEDIATED BY 5-HT1A-RECEPTORS IN THE RAT HIPPOCAMPUS [J].
HOYER, D ;
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ENGEL, G .
EXPERIENTIA, 1986, 42 (06) :637-637
[42]   Regulation of sensitivity to 5-hydroxytryptamine in pulmonary supernumerary but not conventional arteries by a 5-HT1D-like receptor [J].
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Brown, T ;
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TSUJITA, R ;
YAMADA, S ;
SAGAI, H .
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[44]   3-[2-(pyrrolidin-1-yl)ethyl]indoles and analogues: Agonists for the 5-HT1D receptor with high selectivity over the 5-HT1D subtype. [J].
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Guiblin, AR ;
Jelley, R ;
Matassa, VG ;
Russell, MGN ;
Sternfeld, F ;
Beer, M ;
Stanton, J .
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Izzarelli, DG ;
LewisHiggins, L ;
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