STUDIES ON ELECTROGENIC ACTION OF ACETYLCHOLINE WITH TORPEDO-MARMORATA ELECTRIC ORGAN .4. QUINACRINE - FLUORESCENT-PROBE FOR CONFORMATIONAL TRANSITIONS OF CHOLINERGIC RECEPTOR PROTEIN IN ITS MEMBRANE-BOUND STATE

被引:110
作者
GRUNHAGEN, HH [1 ]
CHANGEUX, JP [1 ]
机构
[1] INST PASTEUR,F-75015 PARIS,FRANCE
关键词
D O I
10.1016/0022-2836(76)90249-7
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:497 / 516
页数:20
相关论文
共 25 条
[1]  
Albert A., 1966, ACRIDINES
[2]   USE OF A SNAKE VENON TOXIN TO CHARACTERIZE CHOLINERGIC RECEPTOR PROTEIN [J].
CHANGEUX, JP ;
KASAI, M ;
LEE, CY .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1970, 67 (03) :1241-+
[3]  
COHEN JB, 1972, FEBS LETT, V26, P43, DOI 10.1016/0014-5793(72)80538-6
[4]   INTERACTION OF A FLUORESCENT LIGAND WITH MEMBRANE-BOUND CHOLINERGIC RECEPTOR FROM TORPEDO-MARMORATA [J].
COHEN, JB ;
CHANGEUX, JP .
BIOCHEMISTRY, 1973, 12 (24) :4855-4864
[5]  
COHEN JB, 1974, MOL PHARMACOL, V10, P904
[6]  
ELDEFRAWI M E, 1971, Pesticide Biochemistry and Physiology, V1, P101, DOI 10.1016/0048-3575(71)90215-X
[7]  
GRUNHAGEN H, 1975, CR ACAD SCI D NAT, V281, P1047
[8]   STUDIES ON ELECTROGENIC ACTION OF ACETYLCHOLINE WITH TORPEDO-MARMORATA ELECTRIC ORGAN .5. QUALITATIVE CORRELATION BETWEEN PHARMACOLOGICAL EFFECTS AND EQUILIBRATION PROCESSES OF CHOLINERGIC RECEPTOR PROTEIN AS REVEALED BY STRUCTURAL PROBE QUINACRINE [J].
GRUNHAGEN, HH ;
CHANGEUX, JP .
JOURNAL OF MOLECULAR BIOLOGY, 1976, 106 (03) :517-535
[9]   APPARENT DISSOCIATION CONSTANTS BETWEEN CARBAMYLCHOLINE, DELTA-TUBOCURARINE AND RECEPTOR [J].
HIGMAN, HB ;
PODLESKI, TR ;
BARTELS, E .
BIOCHIMICA ET BIOPHYSICA ACTA, 1963, 75 (02) :187-+