CATECHOL O-METHYLTRANSFERASE .6. AFFINITY LABELING WITH N-HALOACETYL-3,5-DIMETHOXY-4-HYDROXYPHENYLALKYLAMINES

被引：12

作者：

BORCHARDT, RT ^{[1
]}

THAKKER, DR ^{[1
]}

机构：

[1] UNIV KANSAS,DEPT BIOCHEM,MCCOLLUM LABS,LAWRENCE,KS 66044

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1975年 / 18卷 / 02期

关键词：

D O I：

10.1021/jm00236a008

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：152 / 158

页数：7

共 16 条

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[2]

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[3] SYNTHESIS OF 4-HYDROXY-3,5-DIMETHOXY-BETA-PHENETHYLAMINE AND 4-ETHOXY-3,5-DIMETHOXY-BETA-PHENETHYLAMINE [J].

BENINGTON, F ;

MORIN, RD ;

CLARKE, LC .

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[4] CATECHOL ORTHO METHYLTRANSFERASE .4. IN-VITRO INHIBITION BY 3-HYDROXY-4-PYRONES, 3-HYDROXY-2-PYRIDONES, AND 3-HYDROXY-4-PYRIDONES [J].

BORCHARD.RT .

JOURNAL OF MEDICINAL CHEMISTRY, 1973, 16 (05) :581-583

[5] CATECHOL O-METHYLTRANSFERASE .2. IN-VITRO INHIBITION BY SUBSTITUTED 8-HYDROXYQUINOLINES [J].

BORCHARDT, RT .

JOURNAL OF MEDICINAL CHEMISTRY, 1973, 16 (04) :382-387

[6] CATECHOL O-METHYLTRANSFERASE .1. KINETICS OF TROPOLONE INHIBITION [J].

BORCHARDT, RT .

JOURNAL OF MEDICINAL CHEMISTRY, 1973, 16 (04) :377-382

[7] AFFINITY LABELING OF CATECHOL-O-METHYLTRANSFERASE WITH N-IODOACETYL-3,5-DIMETHOXY-4-HYDROXY-PHENYLETHYLAMINE [J].

BORCHARDT, RT ;

THAKKER, D .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1973, 54 (03) :1233-1239

[8] CATECHOL O-METHYLTRANSFERASE .3. MECHANISM OF PYRIDOXAL 5'-PHOSPHATE INHIBITION [J].

BORCHARDT, RT .

JOURNAL OF MEDICINAL CHEMISTRY, 1973, 16 (04) :387-391

[9]

BORCHARDT RT, TO BE PUBLISHED

[10]

BUCK JS, 1943, ORG SYNTH, V2, P622

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