NEUROMEDIN-N - HIGH-AFFINITY INTERACTION WITH BRAIN NEUROTENSIN RECEPTORS AND RAPID INACTIVATION BY BRAIN SYNAPTIC PEPTIDASES

被引:76
作者
CHECLER, F [1 ]
VINCENT, JP [1 ]
KITABGI, P [1 ]
机构
[1] FAC SCI NICE,CTR BIOCHIM,CNRS,F-06034 NICE,FRANCE
关键词
D O I
10.1016/0014-2999(86)90053-1
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:239 / 244
页数:6
相关论文
共 17 条
[1]   DEGRADATION OF NEUROTENSIN BY RAT-BRAIN SYNAPTIC-MEMBRANES - INVOLVEMENT OF A THERMOLYSIN-LIKE METALLOENDOPEPTIDASE (ENKEPHALINASE), ANGIOTENSIN-CONVERTING ENZYME, AND OTHER UNIDENTIFIED PEPTIDASES [J].
CHECLER, F ;
VINCENT, JP ;
KITABGI, P .
JOURNAL OF NEUROCHEMISTRY, 1983, 41 (02) :375-384
[2]   INACTIVATION OF NEUROTENSIN BY RAT-BRAIN SYNAPTIC-MEMBRANES PARTLY OCCURS THROUGH CLEAVAGE AT THE ARG8-ARG9 PEPTIDE-BOND BY A METALLOENDOPEPTIDASE [J].
CHECLER, F ;
VINCENT, JP ;
KITABGI, P .
JOURNAL OF NEUROCHEMISTRY, 1985, 45 (05) :1509-1513
[3]   INACTIVATION OF NEUROTENSIN BY RAT-BRAIN SYNAPTIC-MEMBRANES - CLEAVAGE AT THE PRO10-TYR11 BOND BY ENDOPEPTIDASE-24.11 (ENKEPHALINASE) AND A PEPTIDASE DIFFERENT FROM PROLINE-ENDOPEPTIDASE [J].
CHECLER, F ;
EMSON, PC ;
VINCENT, JP ;
KITABGI, P .
JOURNAL OF NEUROCHEMISTRY, 1984, 43 (05) :1295-1301
[4]   DYNORPHIN1-8 AND DYNORPHIN1-9 ARE LIGANDS FOR THE KAPPA-SUBTYPE OF OPIATE RECEPTOR [J].
CORBETT, AD ;
PATERSON, SJ ;
MCKNIGHT, AT ;
MAGNAN, J ;
KOSTERLITZ, HW .
NATURE, 1982, 299 (5878) :79-81
[5]   DEGRADATION OF CHOLECYSTOKININ-LIKE PEPTIDES BY A CRUDE RAT-BRAIN SYNAPTOSOMAL FRACTION - A STUDY BY HIGH-PRESSURE LIQUID-CHROMATOGRAPHY [J].
DESCHODTLANCKMAN, M ;
BUI, ND ;
NOYER, M ;
CHRISTOPHE, J .
REGULATORY PEPTIDES, 1981, 2 (01) :15-30
[7]   C-FRAGMENT OF BETA-LIPOTROPIN - ENDOGENOUS NEUROLEPTIC OR ANTIPSYCHOTOGEN [J].
JACQUET, YF ;
MARKS, N .
SCIENCE, 1976, 194 (4265) :632-635
[8]   ISOLATION OF SYNAPTIC PLASMA-MEMBRANE FROM BRAIN BY COMBINED FLOTATION-SEDIMENTATION DENSITY GRADIENT CENTRIFUGATION [J].
JONES, DH ;
MATUS, AI .
BIOCHIMICA ET BIOPHYSICA ACTA, 1974, 356 (03) :276-287
[9]   NEUROTENSIN - SPECIFIC BINDING TO SYNAPTIC-MEMBRANES FROM RAT-BRAIN [J].
KITABGI, P ;
CARRAWAY, R ;
VANRIETSCHOTEN, J ;
GRANIER, C ;
MORGAT, JL ;
MENEZ, A ;
LEEMAN, S ;
FREYCHET, P .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1977, 74 (05) :1846-1850
[10]  
KITABGI P, 1980, MOL PHARMACOL, V18, P11