IS TL-99 A SELECTIVE PRE-SYNAPTIC DOPAMINE RECEPTOR AGONIST

被引:53
|
作者
HORN, AS [1 ]
DEVRIES, J [1 ]
DIJKSTRA, D [1 ]
MULDER, AH [1 ]
机构
[1] FREE UNIV AMSTERDAM,DEPT PHARMACOL,1007 MC AMSTERDAM,NETHERLANDS
关键词
D O I
10.1016/0014-2999(82)90283-7
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:35 / 45
页数:11
相关论文
共 50 条
  • [1] ANTIHYPERTENSIVE ACTIVITY OF LY141865, A SELECTIVE PRE-SYNAPTIC DOPAMINE RECEPTOR AGONIST
    HAHN, RA
    MACDONALD, BR
    MARTIN, MA
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 1983, 224 (01): : 206 - 214
  • [2] POSTSYNAPTIC DOPAMINE AGONIST PROPERTIES OF TL-99 ARE REVEALED BY YOHIMBINE CO-TREATMENT
    PASTOR, G
    FALLON, S
    WELCH, JJ
    LIEBMAN, JM
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1983, 87 (04) : 459 - 464
  • [3] METYRAPONE AND SKF 525-A INHIBITION OF A PRE-SYNAPTIC DOPAMINE AGONIST
    KOONS, JC
    FLYNN, JR
    CANNON, JG
    LONG, JP
    FEDERATION PROCEEDINGS, 1982, 41 (05) : 1662 - 1662
  • [4] SK-AND-F-85174 - A DOPAMINE AGONIST WITH PRE-SYNAPTIC ACTIVITY
    BLUMBERG, AL
    HIEBLE, JP
    MCCAFFERTY, J
    HAHN, RA
    SMITH, J
    FEDERATION PROCEEDINGS, 1982, 41 (04) : 1345 - 1345
  • [5] STRUCTURE ACTIVITY RELATIONSHIPS OF PRE-SYNAPTIC DOPAMINE RECEPTOR AGONISTS
    BHATNAGAR, RK
    ARNERIC, SP
    CANNON, JG
    FLYNN, J
    LONG, JP
    PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, 1982, 17 : 11 - 19
  • [6] THE PRE-SYNAPTIC RECEPTOR CONTROVERSY
    KALSNER, S
    TRENDS IN PHARMACOLOGICAL SCIENCES, 1982, 3 (01) : 11 - 21
  • [7] PRE-SYNAPTIC INHIBITION BY DOPAMINE RECEPTOR AGONISTS OF NORADRENERGIC NEUROTRANSMISSION IN THE RABBIT HYPOTHALAMUS
    GALZIN, AM
    DUBOCOVICH, ML
    LANGER, SZ
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 1982, 221 (02): : 461 - 471
  • [8] A COMPARISON OF THE POTENCIES OF VARIOUS DOPAMINE RECEPTOR AGONISTS IN MODELS FOR PRE-SYNAPTIC AND POSTSYNAPTIC RECEPTOR ACTIVITY
    FEENSTRA, MGP
    SUMNERS, C
    GOEDEMOED, JH
    DEVRIES, JB
    ROLLEMA, H
    HORN, AS
    NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1983, 324 (02) : 108 - 115
  • [9] ERGOMETRINE - PRE-SYNAPTIC ALPHA-ADRENOCEPTOR AGONIST
    MARSHALL, I
    NASMYTH, PA
    RUSSELL, GK
    SHEPPERSON, NB
    BRITISH JOURNAL OF PHARMACOLOGY, 1977, 61 (01) : P129 - P129
  • [10] PHARMACOLOGICAL PROFILES OF THE PUTATIVE DOPAMINE AUTORECEPTOR AGONISTS 3-PPP AND TL-99
    MARTIN, GE
    HAUBRICH, DR
    WILLIAMS, M
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 76 (01) : 15 - 23