COMPARISON OF THE BETA-1-SELECTIVE AFFINITY OF PRENALTEROL AND CORWIN DEMONSTRATED BY RADIOLIGAND BINDING

被引:37
作者
COOK, N [1 ]
RICHARDSON, A [1 ]
BARNETT, DB [1 ]
机构
[1] UNIV LEICESTER,LEICESTER ROYAL INFIRM,DEPT PHARMACOL & THERAPEUT,LEICESTER LE2 7LX,ENGLAND
关键词
D O I
10.1016/0014-2999(84)90289-9
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:407 / 412
页数:6
相关论文
共 17 条
[1]   PRENALTEROL IS AN AGONIST AT BETA-2-ADRENOCEPTOR AS WELL AS AT BETA-1-ADRENOCEPTORS [J].
APPERLEY, GH ;
DREW, GM ;
SULLIVAN, AT .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 81 (04) :659-663
[2]   DIFFERENTIATION OF CARDIAC CHRONOTROPIC AND INOTROPIC EFFECTS OF BETA-ADRENOCEPTOR AGONISTS [J].
CARLSSON, E ;
DAHLOF, CG ;
HEDBERG, A ;
PERSSON, H ;
TANGSTRAND, B .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1977, 300 (02) :101-105
[3]  
COHEN ML, 1980, J PHARMACOL EXP THER, V215, P325
[4]   SIMULTANEOUS ANALYSIS OF FAMILIES OF SIGMOIDAL CURVES - APPLICATION TO BIOASSAY, RADIOLIGAND ASSAY, AND PHYSIOLOGICAL DOSE-RESPONSE CURVES [J].
DELEAN, A ;
MUNSON, PJ ;
RODBARD, D .
AMERICAN JOURNAL OF PHYSIOLOGY, 1978, 235 (02) :E97-E102
[5]   PRENALTEROL, A NON-SELECTIVE BETA-ADRENOCEPTOR LIGAND WITH ABSOLUTE BETA-1-SELECTIVE PARTIAL AGONIST ACTIVITY [J].
HEDBERG, A ;
MATTSSON, H ;
CARLSSON, E .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1980, 32 (09) :660-661
[6]  
KENAKIN TP, 1982, J PHARMACOL EXP THER, V223, P416
[7]  
KENAKIN TP, 1980, J PHARMACOL EXP THER, V213, P406
[8]  
KENAKIN TP, 1982, J PHARMACOL EXP THER, V220, P77
[9]  
KENT RS, 1980, MOL PHARMACOL, V17, P14
[10]   BETA-1-ADRENOCEPTOR AND BETA-2-ADRENOCEPTOR STIMULATORY EFFECTS OF PRENALTEROL [J].
MATTSSON, H ;
ANDERSSON, T ;
CARLSSON, E ;
HEDBERG, A ;
LUNDGREN, B ;
OLSSON, T .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1982, 321 (04) :302-308