AVERMECTIN B1A INHIBITS THE BINDING OF STRYCHNINE TO THE GLYCINE RECEPTOR OF RAT SPINAL-CORD

被引:37
作者
GRAHAM, D [1 ]
PFEIFFER, F [1 ]
BETZ, H [1 ]
机构
[1] MAX PLANCK INST PSYCHIAT,DEPT NEUROCHEM,D-8033 MARTINSRIED,FED REP GER
关键词
D O I
10.1016/0304-3940(82)90349-4
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:173 / 176
页数:4
相关论文
共 12 条
[1]  
CURTIS DR, 1968, EXP BRAIN RES, V5, P235
[2]   AVERMECTIN-B1A IRREVERSIBLY BLOCKS POSTSYNAPTIC POTENTIALS AT THE LOBSTER NEUROMUSCULAR-JUNCTION BY REDUCING MUSCLE MEMBRANE RESISTANCE [J].
FRITZ, LC ;
WANG, CC ;
GORIO, A .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1979, 76 (04) :2062-2066
[3]   STEREOSPECIFIC INTERACTION OF BICUCULLINE WITH SPECIFIC [STRYCHNINE-H-3 BINDING TO RAT SPINAL-CORD SYNAPTOSOMAL MEMBRANES [J].
GOLDINGER, A ;
MULLER, WE .
NEUROSCIENCE LETTERS, 1980, 16 (01) :91-95
[4]   UV LIGHT-INDUCED CROSS-LINKING OF STRYCHNINE TO THE GLYCINE RECEPTOR OF RAT SPINAL-CORD MEMBRANES [J].
GRAHAM, D ;
PFEIFFER, F ;
BETZ, H .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1981, 102 (04) :1330-1335
[5]   GABA-BENZODIAZEPINE-BARBITURATE RECEPTOR INTERACTIONS [J].
OLSEN, RW .
JOURNAL OF NEUROCHEMISTRY, 1981, 37 (01) :1-13
[6]   AVERMECTIN B1A - AN IRREVERSIBLE ACTIVATOR OF THE GAMMA-AMINOBUTYRIC ACID-BENZODIAZEPINE-CHLORIDE-IONOPHORE RECEPTOR COMPLEX [J].
PAUL, SM ;
SKOLNICK, P ;
ZATZ, M .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1980, 96 (02) :632-638
[7]   SOLUBILIZATION OF THE GLYCINE RECEPTOR FROM RAT SPINAL-CORD [J].
PFEIFFER, F ;
BETZ, H .
BRAIN RESEARCH, 1981, 226 (1-2) :273-279
[8]   SPECIFICITY OF HIGH-AFFINITY BINDING OF AVERMECTIN-B1A TO MAMMALIAN BRAIN [J].
PONG, SS ;
WANG, CC .
NEUROPHARMACOLOGY, 1980, 19 (03) :311-317
[9]   INVITRO MODULATION BY AVERMECTIN-B1A OF THE GABA-BENZODIAZEPINE RECEPTOR COMPLEX OF RAT CEREBELLUM [J].
SUPAVILAI, P ;
KAROBATH, M .
JOURNAL OF NEUROCHEMISTRY, 1981, 36 (03) :798-803
[10]   ENHANCEMENT OF INVITRO BINDING AND SOME OF THE PHARMACOLOGICAL PROPERTIES OF DIAZEPAM BY A NOVEL ANTHELMINTIC AGENT, AVERMECTIN-B1A [J].
WILLIAMS, M ;
YARBROUGH, GG .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1979, 56 (03) :273-276