ANTAGONISM OF 5-HYDROXYTRYPTAMINE1A (5-HT1A) RECEPTOR-MEDIATED MODULATION OF ADENYLATE-CYCLASE ACTIVITY BY PINDOLOL AND PROPRANOLOL ISOMERS

被引:71
作者
OKSENBERG, D
PEROUTKA, SJ
机构
[1] STANFORD UNIV,DEPT NEUROL,STANFORD,CA 94305
[2] STANFORD UNIV,DEPT PHARMACOL,STANFORD,CA 94305
关键词
D O I
10.1016/0006-2952(88)90692-2
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:3429 / 3433
页数:5
相关论文
共 31 条
[21]  
PEROUTKA SJ, 1979, MOL PHARMACOL, V16, P687
[22]   ROLE OF HORMONE RECEPTORS AND GTP-REGULATORY PROTEINS IN MEMBRANE TRANSDUCTION [J].
RODBELL, M .
NATURE, 1980, 284 (5751) :17-22
[23]  
Salomon Y, 1979, Adv Cyclic Nucleotide Res, V10, P35
[24]   NUCLEOTIDE INTERACTIONS WITH 5-HT1A BINDING-SITES DIRECTLY LABELED BY [H-3] 8-HYDROXY-2-(DI-NORMAL-PROPYLAMINO)TETRALIN ([H-3]-8-OH-DPAT) [J].
SCHLEGEL, JR ;
PEROUTKA, SJ .
BIOCHEMICAL PHARMACOLOGY, 1986, 35 (12) :1943-1949
[25]   MESSAGE TRANSMISSION - RECEPTOR CONTROLLED ADENYLATE-CYCLASE SYSTEM [J].
SCHRAMM, M ;
SELINGER, Z .
SCIENCE, 1984, 225 (4668) :1350-1356
[26]   FORSKOLIN, CYCLIC-AMP AND CELLULAR PHYSIOLOGY [J].
SEAMON, KB ;
DALY, JW .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1983, 4 (03) :120-123
[27]   FORSKOLIN - UNIQUE DITERPENE ACTIVATOR OF ADENYLATE-CYCLASE IN MEMBRANES AND IN INTACT-CELLS [J].
SEAMON, KB ;
PADGETT, W ;
DALY, JW .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1981, 78 (06) :3363-3367
[28]  
SHENKER A, 1983, LIFE SCI, V32, P2335, DOI 10.1016/0024-3205(83)90763-4
[29]  
SPROUSE JS, 1987, EUR J PHARM, V128, P713
[30]  
TRICKLEBANK MD, 1985, EUROPEAN J PHARM, V106, P271