MOLECULAR THEORY OF DRUG ACTION BASED ON INDUCED CONFORMATIONAL PERTURBATIONS OF RECEPTORS

被引:145
作者
BELLEAU, B
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D O I
10.1021/jm00336a022
中图分类号
R914 [药物化学];
学科分类号
100701 ;
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页码:776 / &
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[1]   MOLECULAR BASIS FOR DRUG ACTION [J].
ARIENS, EJ ;
SIMONIS, AM .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1964, 16 (03) :137-&
[2]  
ARIENS EJ, 1954, ARCH INT PHARMACOD T, V99, P32
[3]  
ARIENS EJ, 1956, ARZNEIMITTEL-FORSCH, V6, P282
[4]   MOLECULAR BASIS FOR DRUG ACTION . INTERACTION OF 1 OR MORE DRUGS WITH DIFFERENT RECEPTORS [J].
ARIENS, EJ ;
SIMONIS, AM .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1964, 16 (05) :289-&
[5]  
ARIENS EJ, 1957, PHARMACOL REV, V9, P218
[6]   AN ATTEMPT TO STUDY EFFECTS OF CHEMICAL STRUCTURE ON AFFINITY AND EFFICACY OF COMPOUNDS RELATED TO ACETYLCHOLINE [J].
BARLOW, RB ;
SCOTT, KA ;
STEPHENSON, RP .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1963, 21 (03) :509-&
[7]  
BECKETT AH, 1962, 1 P INT PHARM M STOC, V7, P28
[8]  
BECKETT AH, 1962, 1 P INT PHARM M STOC, V7, P31
[9]   STEREOCHEMISTRY OF INTERACTION OF ENANTIOMETIC 1,3-DIOXOLANE ANALOGS OF MUSCARONE WITH CHOLINERGIC RECEPTORS [J].
BELLEAU, B ;
PURANEN, J .
JOURNAL OF MEDICINAL CHEMISTRY, 1963, 6 (03) :325-&
[10]   ASPECTS OF CHEMICAL MECHANISM OF COMPLEX FORMATION BETWEEN ACETYLCHOLINESTERASE + ACETYLCHOLINE-RELATED COMPOUNDS [J].
BELLEAU, B ;
LACASSE, G .
JOURNAL OF MEDICINAL CHEMISTRY, 1964, 7 (06) :768-&