CONVERSION OF DOPAMINE-D1 RECEPTORS FROM HIGH TO LOW AFFINITY FOR DOPAMINE

被引：102

作者：

SEEMAN, P ^{[1
]}

ULPIAN, C ^{[1
]}

GRIGORIADIS, D ^{[1
]}

PRIBAR, I ^{[1
]}

BUCHMAN, O ^{[1
]}

机构：

[1] NUCL RES CTR NEGEV,DEPT BIOCHEM,IL-84190 BEERSHEBA,ISRAEL

来源：

BIOCHEMICAL PHARMACOLOGY | 1985年 / 34卷 / 01期

关键词：

D O I：

10.1016/0006-2952(85)90116-9

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：151 / 154

页数：4

共 19 条

[1] CHARACTERISTICS OF CIS-FLUPENTHIXOL-H-3 BINDING TO CALF BRAIN MEMBRANES [J].

CROSS, AJ ;

OWEN, F .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1980, 65 (04) :341-347

[2]

GEORGE SR, 1983, DOPAMINE RECEPTORS, P93

[3]

GOLDBERG LI, 1979, COMMUN PSYCHOPHARMAC, V3, P447

[4] THE DOPAMINE NEUROLEPTIC RECEPTOR [J].

GRIGORIADIS, D ;

SEEMAN, P .

CANADIAN JOURNAL OF NEUROLOGICAL SCIENCES, 1984, 11 (01) :108-113

[5] H-3-DOPAMINE BINDING TO RAT STRIATAL D-2 AND D-3 SITES - ENHANCEMENT BY MAGNESIUM AND INHIBITION BY GUANINE-NUCLEOTIDES AND SODIUM [J].

HAMBLIN, MW ;

CREESE, I .

LIFE SCIENCES, 1982, 30 (18) :1587-1595

[6] SCH-23390 - THE 1ST SELECTIVE DOPAMINE D-1 ANTAGONIST [J].

HYTTEL, J .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1983, 91 (01) :153-154

[7] COMPARISON OF EFFECT OF NEUROLEPTIC DRUGS ON BINDING OF HALOPERIDOL-H-3 AND CIS(Z)-FLUPENTHIXOL-H-3 AND ON ADENYLATE-CYCLASE ACTIVITY IN RAT STRIATAL TISSUE INVITRO [J].

HYTTEL, J .

PROGRESS IN NEURO-PSYCHOPHARMACOLOGY, 1978, 2 (03) :329-335

[8]

IORIO LC, 1983, J PHARMACOL EXP THER, V226, P462

[9] MULTIPLE RECEPTORS FOR DOPAMINE [J].

KEBABIAN, JW ;

CALNE, DB .

NATURE, 1979, 277 (5692) :93-96

[10] DOPAMINE-RECEPTORS RE-EXPLAINED [J].

LEFF, SE ;

CREESE, I .

TRENDS IN PHARMACOLOGICAL SCIENCES, 1983, 4 (11) :463-467

← 1 2 →