SYNTHESIS AND BIOLOGICAL-ACTIVITIES OF DYNORPHIN-A ANALOGS WITH OPIOID ANTAGONIST PROPERTIES

被引：27
作者：
GAIRIN, JE [1 ]
MAZARGUIL, H [1 ]
ALVINERIE, P [1 ]
SAINTPIERRE, S [1 ]
MEUNIER, JC [1 ]
CROS, J [1 ]
机构：
[1] UNIV SHERBROOKE,FAC MED,DEPT PHYSIOL & PHARMACOL,SHERBROOKE J1H 5N4,QUEBEC,CANADA
来源：
JOURNAL OF MEDICINAL CHEMISTRY | 1986年 / 29卷 / 10期
关键词：
D O I：
10.1021/jm00160a019
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
引用
收藏
页码：1913 / 1917
页数：5
相关论文
共 39 条
  • [11] [D-PRO(10)]DYNORPHIN-(1-11) IS A HIGHLY POTENT AND SELECTIVE LIGAND FOR KAPPA-OPIOID RECEPTORS
    GAIRIN, JE
    GOUARDERES, C
    MAZARGUIL, H
    ALVINERIE, P
    CROS, J
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 106 (02) : 457 - 458
  • [12] MONITORING OF REACTIONS IN SOLID-PHASE PEPTIDE SYNTHESIS WITH PICRIC ACID
    GISIN, BF
    [J]. ANALYTICA CHIMICA ACTA, 1972, 58 (01) : 248 - &
  • [13] PREPARATION OF MERRIFIELD-RESINS THROUGH TOTAL ESTERIFICATION WITH CESIUM SALTS
    GISIN, BF
    [J]. HELVETICA CHIMICA ACTA, 1973, 56 (05) : 1476 - 1482
  • [14] PORCINE PITUITARY DYNORPHIN - COMPLETE AMINO-ACID-SEQUENCE OF THE BIOLOGICALLY-ACTIVE HEPTADECAPEPTIDE
    GOLDSTEIN, A
    FISCHLI, W
    LOWNEY, LI
    HUNKAPILLER, M
    HOOD, L
    [J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1981, 78 (11): : 7219 - 7223
  • [15] GOLDSTEIN A, 1984, MECHANISM DRUG ACTIO, P49
  • [16] IMMUNOREACTIVE DYNORPHIN IN HUMAN-BRAIN AND PITUITARY
    GRAMSCH, C
    HOLLT, V
    PASI, A
    MEHRAEIN, P
    HERZ, A
    [J]. BRAIN RESEARCH, 1982, 233 (01) : 65 - 74
  • [17] AGONIST AND ANTAGONIST ACTIONS OF MORPHINE-LIKE DRUGS ON GUINEA-PIG ISOLATED ILEUM
    GYANG, EA
    KOSTERLITZ, HW
    [J]. BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1966, 27 (03): : 514 - +
  • [18] ANALOGS OF BETA-LPH61-64 POSSESSING SELECTIVE AGONIST ACTIVITY AT MU-OPIATE RECEPTORS
    HANDA, BK
    LANE, AC
    LORD, JAH
    MORGAN, BA
    RANCE, MJ
    SMITH, CFC
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 70 (04) : 531 - 540
  • [19] ANTI-NOCICEPTIVE PROFILE OF DYNORPHIN IN THE RAT
    HAYES, AG
    SKINGLE, M
    TYERS, MB
    [J]. LIFE SCIENCES, 1983, 33 : 657 - 660
  • [20] JAMES IF, 1984, J PHARMACOL EXP THER, V228, P88
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