REGIOSELECTIVE ADAMANTYLATION OF N-UNSUBSTITUTED PYRAZOLE DERIVATIVES

被引：14
作者：
CABILDO, P
CLARAMUNT, RM
FORFAR, I
ELGUERO, J
机构：
[1] Univ Nacl Educ Distancia, DEPT QUIM ORGAN & BIOL, E-28040 MADRID, SPAIN
[2] Univ Nacl Educ Distancia, INST QUIM MED, E-28040 MADRID, SPAIN
[3] CSIC, E-28040 MADRID, SPAIN
来源：
TETRAHEDRON LETTERS | 1994年 / 35卷 / 01期
关键词：
D O I：
10.1016/0040-4039(94)88196-0
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Reaction of NH-pyrazoles with 1-bromoadamantane in a high pressure stainless steel autoclave (250 ml, maximum working pressure of 200 atm) gives regioselectively 1-adamantyl or 4-adamantylpyrazoles depending on the temperature.
引用
收藏
页码：183 / 184
页数：2
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