DESIGN AND SYNTHESIS OF 5,6-DIHYDRO-4H-1,3,4-OXADIAZINES AS POTENTIAL OCTOPAMINERGIC INSECTICIDES

被引：17

作者：

DEKEYSER, MA

HARRISON, WA

MCDONALD, PT

DOWNER, RGH

机构：

[1] UNIROYAL CHEM INC,NEW PROD RES,BETHANY,CT 06525

[2] UNIV WATERLOO,DEPT BIOL,WATERLOO N2L 3G1,ONTARIO,CANADA

来源：

PESTICIDE SCIENCE | 1993年 / 38卷 / 04期

关键词：

D O I：

10.1002/ps.2780380405

中图分类号：

S3 [农学（农艺学）];

学科分类号：

0901 ;

摘要：

A novel class of insecticides, the dihydrooxadiazines, was proposed following the use of molecular modelling techniques. These compounds represent conformationally restricted analogues of octopamine. Eight dihydrooxadiazines were synthesized and evaluated for useful insecticidal properties. Several of these compounds demonstrated activity against rice planthoppers, mite eggs, and tobacco budworm eggs.

引用

页码：309 / 314

页数：6

共 12 条

[1]

DOWNER RGH, 1990, COCKROACHES MODELS N, V11, P103

[2]

DOWNER RGH, 1988, MOL BASIS DRUG PESTI, P255

[3]

Evans P.D., 1980, Advances in Insect Physiology, V15, P317, DOI 10.1016/S0065-2806(08)60143-5

[4]

Evans P.D., 1985, P499