CONCENTRATION-EFFECT RELATIONSHIPS WITH FM-24 - A NEW LONG-ACTING BETA-ADRENERGIC-RECEPTOR ANTAGONIST

被引:7
作者
DOLLERY, CT [1 ]
DARGIE, HJ [1 ]
SASSARD, J [1 ]
CUISINAUD, G [1 ]
机构
[1] FAC PHARM LYON,DEPT PHYSIOL & PHARMACOL CLIN,CNRS,ERA 894,F-69008 LYON,FRANCE
关键词
D O I
10.1111/j.1365-2125.1983.tb01554.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:707 / 713
页数:7
相关论文
共 20 条
[1]   SENSITIVE GAS-CHROMATOGRAPHIC METHOD FOR THE DETERMINATION IN PLASMA OF FM 24,1-(2-EXO-BICYCLO[2,2,1]HEPT-2-YLPHENOXY)-3-[(1-METHYLETHYL)AMINO]-2-PROPANOL, A NEW BETA-ADRENOCEPTOR BLOCKING-AGENT [J].
BERNARD, N ;
CUISINAUD, G ;
JOZEFCZAK, C ;
SECCIA, M ;
FERRY, N ;
SASSARD, J .
JOURNAL OF CHROMATOGRAPHY, 1980, 183 (01) :99-103
[2]   PLASMA PROPRANOLOL LEVELS IN QUANTITATIVE ASSESSMENT OF BETA-ADRENERGIC BLOCKADE IN MAN [J].
COLTART, DJ ;
SHAND, DG .
BRITISH MEDICAL JOURNAL, 1970, 3 (5725) :731-&
[3]   POTENTIAL PROBE FOR ISOLATION OF BETA-ADRENOCEPTOR, CHLOROPRACTOLOL [J].
EREZ, M ;
WEINSTOCK, M ;
COHEN, S ;
SHTACHER, G .
NATURE, 1975, 255 (5510) :635-636
[4]   THE SYNTHESIS OF BETA-ADRENERGIC RECEPTORS IN CULTURED HUMAN-LUNG CELLS - INDUCTION BY GLUCOCORTICOIDS [J].
FRASER, CM ;
VENTER, JC .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1980, 94 (01) :390-397
[5]  
GEORGE CF, 1973, BIOLOGICAL EFFECTS D, P123
[6]  
GOLDSTEIN A, 1974, PRINCIPLES DRUG ACTI
[7]   MUSCLE-ACTIVITY DECREASES RATE OF DEGRADATION OF ALPHA-BUNGAROTOXIN BOUND TO EXTRAJUNCTIONAL ACETYLCHOLINE RECEPTORS [J].
HOGAN, PG ;
MARSHALL, JM ;
HALL, ZW .
NATURE, 1976, 261 (5558) :328-330
[8]  
JONES GR, 1981, BRIT HEART J, V46, P503
[9]   CAN CHLOROPRACTOLOL ALKYLATE BETA-ADRENOCEPTORS [J].
KENAKIN, TP ;
BLACK, JW .
NATURE, 1977, 265 (5592) :365-366
[10]  
KENT RS, 1980, MOL PHARMACOL, V17, P14