SYNTHESIS AND CHARACTERIZATION OF 2-HYDROXYMETHYL-1-METHYL-4-NITRO-5-IMIDAZOLCARBONITRILE-4,5-14C

被引：0

作者：

ELLSWORTH, RL

MERIWETHER, HT

MERTEL, HE

机构：

[1] Merck Sharp & Dohme Research Laboratories, Rahway, New Jersey, 07065

来源：

JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS | 1990年 / 28卷 / 07期

关键词：

D O I：

10.1002/jlcr.2580280702

中图分类号：

Q5 [生物化学];

学科分类号：

071010 ; 081704 ;

摘要：

Preparation of the title compound, a key intermediate required to assist in the investigation and development of a new class of substances for controlling coccidiosis, is described. This labeled substance was synthesized in 10 steps, with a 17% overall radiochemical yield, from oxalic‐1,2‐14C acid. Copyright © 1990 John Wiley & Sons, Ltd.

引用

页码：745 / 751

页数：7

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