ANTI-TUMOR ACTIVITY OF CLOMIPHENE ANALOGS INVITRO - RELATIONSHIP TO AFFINITY FOR THE ESTROGEN-RECEPTOR AND ANOTHER HIGH-AFFINITY ANTIESTROGEN-BINDING SITE

被引：49
作者：
MURPHY, LC [1 ]
SUTHERLAND, RL [1 ]
机构：
[1] UNIV SYDNEY, LUDWIG INST CANC RES, SYDNEY, NSW 2006, AUSTRALIA
来源：
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM | 1983年 / 57卷 / 02期
关键词：
D O I：
10.1210/jcem-57-2-373
中图分类号：
R5 [内科学];
学科分类号：
1002 ; 100201 ;
摘要：
引用
收藏
页码：373 / 379
页数：7
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共 42 条
[21]   ESTRADIOL INHIBITS TRANSCRIPTION OF THE HUMAN GLYCOPROTEIN HORMONE ALPHA-SUBUNIT GENE DESPITE THE ABSENCE OF A HIGH-AFFINITY BINDING-SITE FOR ESTROGEN-RECEPTOR [J].
KERI, RA ;
ANDERSEN, B ;
KENNEDY, GC ;
HAMERNIK, DL ;
CLAY, CM ;
BRACE, AD ;
NETT, TM ;
NOTIDES, AC ;
NILSON, JH .
MOLECULAR ENDOCRINOLOGY, 1991, 5 (05) :725-733
[22]   2-PHENYLINDOLES - RELATIONSHIP BETWEEN STRUCTURE, ESTROGEN-RECEPTOR AFFINITY, AND MAMMARY-TUMOR INHIBITING ACTIVITY IN THE RAT [J].
VONANGERER, E ;
PREKAJAC, J ;
STROHMEIER, J .
JOURNAL OF MEDICINAL CHEMISTRY, 1984, 27 (11) :1439-1447
[23]   52-ANDROSTANE-3-BETA, 17-BETA-DIOL - ANDROGEN WITH HIGH-AFFINITY BINDING FOR CYTOSOLIC ESTROGEN-RECEPTOR [J].
THIEULANT, ML ;
SAMPEREZ, S ;
JOUAN, P .
CANCER TREATMENT REPORTS, 1979, 63 (07) :1162-1162
[24]   A HIGH-AFFINITY BINDING-SITE FOR THE ANTIESTROGENS, TAMOXIFEN AND C1 628, IN IMMATURE RAT UTERINE CYTOSOL WHICH IS DISTINCT FROM THE ESTROGEN-RECEPTOR [J].
MURPHY, LC ;
SUTHERLAND, RL .
JOURNAL OF ENDOCRINOLOGY, 1981, 91 (01) :155-161
[25]   11-BETA-SUBSTITUTED ESTRADIOL DERIVATIVES, POTENTIAL HIGH-AFFINITY CARBON-11-LABELED PROBES FOR THE ESTROGEN-RECEPTOR - A STRUCTURE-AFFINITY RELATIONSHIP STUDY [J].
NAPOLITANO, E ;
FIASCHI, R ;
CARLSON, KE ;
KATZENELLENBOGEN, JA .
JOURNAL OF MEDICINAL CHEMISTRY, 1995, 38 (03) :429-434
[26]   HIGH-AFFINITY BINDING OF ANTI-ESTROGEN [TAMOXIFEN-H-3 TO 8S ESTRADIOL RECEPTOR [J].
CAPONY, F ;
ROCHEFORT, H .
MOLECULAR AND CELLULAR ENDOCRINOLOGY, 1978, 11 (02) :181-198
[27]   NEW HALOGENATED ESTROGENS WITH HIGH BINDING-AFFINITY AND SELECTIVITY FOR THE ESTROGEN-RECEPTOR - POTENTIAL BREAST-TUMOR IMAGING AGENTS [J].
KATZENELLENBOGEN, JA ;
SENDEROFF, SG ;
LANDVATTER, SW ;
MCELVANY, KD ;
WELCH, MJ .
JOURNAL OF NUCLEAR MEDICINE, 1981, 22 (06) :P20-P20
[28]   HIGH-AFFINITY BINDING OF ESTROGEN-RECEPTOR TO RECOMBINANT PLASMIDS CONTAINING (DA-DC)N.(DG-DT)N SEQUENCES [J].
THOMAS, T ;
THOMAS, TJ .
CANCER RESEARCH, 1989, 49 (17) :4734-4739
[29]   [I-125] 17-ALPHA-LODOVINYL 11-BETA-METHOXYESTRADIOL - INVIVO AND INVITRO PROPERTIES OF A HIGH-AFFINITY ESTROGEN-RECEPTOR RADIOPHARMACEUTICAL [J].
JAGODA, EM ;
GIBSON, RE ;
GOODGOLD, H ;
FERREIRA, N ;
FRANCIS, BE ;
REBA, RC ;
RZESZOTARSKI, WJ ;
ECKELMAN, WC .
JOURNAL OF NUCLEAR MEDICINE, 1984, 25 (04) :472-477
[30]   11-BETA-ETHYL-17-ALPHA-ETHYNYLESTRADIOL (EEE2) - INVITRO AND INVIVO CHARACTERIZATION OF A VERY HIGH-AFFINITY ESTROGEN-RECEPTOR RADIOTRACER [J].
SHOOK, MA ;
GIBSON, RE ;
FERREIRA, NL ;
RZESZOTARSKI, WJ ;
REBA, RC .
JOURNAL OF NUCLEAR MEDICINE, 1986, 27 (06) :916-916
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