Synthesis and Characterization of Some Fluorinated 1, 5-Benzothiazepines and Pyrazolines

被引：4

作者：

Jagadhani, S. G. ^{[1
]}

Kundlikar, S. G. ^{[1
]}

Karale, B. K. ^{[1
]}

机构：

[1] Radhabai Kale Mahila Mahavidyalaya, Dept Chem, Ahmednagar 414001, India

来源：

ORIENTAL JOURNAL OF CHEMISTRY | 2015年 / 31卷 / 01期

关键词：

Benzothiazepines; Fluorinated chalcones; Pyrazolines;

D O I：

10.13005/ojc/310177

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

4-Bromo-2-fluorobenzaidehyde 1 when treated with substituted hydroxy acetophenones 2 yields chalcones 3. These chalcones were refluxed with 2-aminothiophenol gave "2-[2-(4-, bromo-2-fluorophenyl)-2,3-dihydro-1,5-benzothiazepin-4-Aphenol" 4 and when treated with hydrazine hydrate gave the compound "2-[5-(4-bromo-2-fluorophenyl)-4,5-dihydro-1H-pyrazol-3-yljphenol" 5. The structures of compounds have been established on the basis of spectral data.

引用

页码：601 / 604

页数：4

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