SOLID-PHASE SYNTHESIS OF VINYLOGOUS SULFONYL PEPTIDES

被引：53

作者：

GENNARI, C

NESTLER, HP

SALOM, B

STILL, WC

机构：

[1] COLD SPRING HARBOR LAB,COLD SPRING HARBOR,NY 11724

[2] COLUMBIA UNIV,DEPT CHEM,NEW YORK,NY 10027

来源：

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH | 1995年 / 34卷 / 16期

关键词：

COMBINATORIAL CHEMISTRY; PEPTIDES; SOLID-PHASE SYNTHESIS; SULFONAMIDES;

D O I：

10.1002/anie.199517631

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Now available for combinatorial compound libraries, vinylogous sulfonyl peptides like 1 may have potential as components of enzyme inhibitors. Newly developed solid‐phase synthesis of these compounds (shown schematically below) opens up these possibilities. • = polyoxyethylene‐grafted crosslinked polystyrene resin. (Figure Presented.) Copyright © 1995 by VCH Verlagsgesellschaft mbH, Germany

引用

页码：1763 / 1765

页数：3

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