RELATIONSHIPS BETWEEN STRUCTURE AND DURATION OF NEUROTENSINS CENTRAL ACTION - EMERGENCE OF LONG-ACTING ANALOGS

被引:26
作者
JOLICOEUR, FB [1 ]
STPIERRE, S [1 ]
AUBE, C [1 ]
RIVEST, R [1 ]
GAGNE, MA [1 ]
机构
[1] UNIV SHERBROOKE,FAC MED,DEPT PHYSIOL & PHARMACOL,SHERBROOKE J1H 5N4,QUEBEC,CANADA
关键词
D O I
10.1016/0143-4179(84)90090-8
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:467 / 476
页数:10
相关论文
共 17 条
[1]  
[Anonymous], 1971, STAT PRINCIPLES EXPT
[2]   DEGRADATION OF NEUROTENSIN BY RAT-BRAIN SYNAPTIC-MEMBRANES - INVOLVEMENT OF A THERMOLYSIN-LIKE METALLOENDOPEPTIDASE (ENKEPHALINASE), ANGIOTENSIN-CONVERTING ENZYME, AND OTHER UNIDENTIFIED PEPTIDASES [J].
CHECLER, F ;
VINCENT, JP ;
KITABGI, P .
JOURNAL OF NEUROCHEMISTRY, 1983, 41 (02) :375-384
[3]  
CHECLER F, 1983, J PHARMACOL EXP THER, V227, P743
[4]   SEIZURES IN RATS ASSOCIATED WITH DIVALENT CATION INHIBITION OF NA+-K+-ATPASE [J].
DONALDSON, J ;
STPIERRE, T ;
MINNICH, J ;
BARBEAU, A .
CANADIAN JOURNAL OF BIOCHEMISTRY, 1971, 49 (11) :1217-+
[5]   ENZYMIC INACTIVATION OF NEUROTENSIN BY HYPOTHALAMIC AND BRAIN EXTRACTS OF RAT [J].
DUPONT, A ;
MERAND, Y .
LIFE SCIENCES, 1978, 22 (18) :1623-1630
[6]   THE REGIONAL DISTRIBUTION AND CHROMATOGRAPHIC CHARACTERIZATION OF NEUROTENSIN-LIKE IMMUNOREACTIVITY IN THE RAT CENTRAL NERVOUS-SYSTEM [J].
EMSON, PC ;
GOEDERT, M ;
HORSFIELD, P ;
RIOUX, F ;
STPIERRE, S .
JOURNAL OF NEUROCHEMISTRY, 1982, 38 (04) :992-999
[7]   DIFFERENTIAL NEURO-BEHAVIORAL EFFECTS OF NEUROTENSIN AND STRUCTURAL ANALOGS [J].
JOLICOEUR, FB ;
BARBEAU, A ;
RIOUX, F ;
QUIRION, R ;
STPIERRE, S .
PEPTIDES, 1981, 2 (02) :171-175
[8]  
JOLICOEUR FB, 1982, BRAIN NEUROTRANSMITT, P171
[9]  
JOLICOEUR FB, 1984, HDB NEUROCHEMISTRY
[10]  
KITABGI P, 1980, MOL PHARMACOL, V18, P11