THE SYNTHESIS OF PHOSPHONATE ANALOGS OF AMINO-ACIDS AND PEPTIDES

被引：0
作者：
HAMILTON, R
KAY, G
SHUTE, RE
TRAVERS, J
WALKER, B
WALKER, BJ
机构：
[1] QUEENS UNIV BELFAST,SCH BIOL SCI,BELFAST BT7 1NN,ANTRIM,NORTH IRELAND
[2] ICI PLC,PHARMACEUT,LONDON,ENGLAND
来源：
PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS | 1993年 / 76卷 / 1-4期
关键词：
D O I：
暂无
中图分类号：
O61 [无机化学];
学科分类号：
070301 ; 081704 ;
摘要：
Diphenyl phosphonate ester analogues of phenylalanine and peptides derived from these have been prepared and are shown to specifically inhibit chymotrypsin. Phosphonate isosters of serine and tyrosine phosphates appropriately protected for use in peptide synthesis have been prepared.
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页码：387 / 390
页数：4
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