NORBINALTORPHIMINE - ANTAGONIST PROFILE AT KAPPA-OPIOID RECEPTORS

被引:92
作者
BIRCH, PJ
HAYES, AG
SHEEHAN, MJ
TYERS, MB
机构
关键词
D O I
10.1016/0014-2999(87)90397-9
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
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页码:405 / 408
页数:4
相关论文
共 10 条
[1]   SOME QUANTITATIVE USES OF DRUG ANTAGONISTS [J].
ARUNLAKSHANA, O ;
SCHILD, HO .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (01) :48-58
[2]  
BIRCH PJ, IN PRESS BR J PHARM
[3]   ICI-174864 - A HIGHLY SELECTIVE ANTAGONIST FOR THE OPIOID DELTA-RECEPTOR [J].
COTTON, R ;
GILES, MG ;
MILLER, L ;
SHAW, JS ;
TIMMS, D .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 97 (3-4) :331-332
[4]  
FINNEY DJ, 1964, STATISTICAL METHODS
[5]   PROFILE OF ACTIVITY OF KAPPA-RECEPTOR AGONISTS IN THE RABBIT VAS-DEFERENS [J].
HAYES, A ;
KELLY, A .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 110 (03) :317-322
[6]   DETERMINATION OF THE RECEPTOR SELECTIVITY OF OPIOID AGONISTS IN THE GUINEA-PIG ILEUM AND MOUSE VAS-DEFERENS BY USE OF BETA-FUNALTREXAMINE [J].
HAYES, AG ;
SHEEHAN, MJ ;
TYERS, MB .
BRITISH JOURNAL OF PHARMACOLOGY, 1985, 86 (04) :899-904
[7]   BINALTORPHIMINE AND NOR-BINALTORPHIMINE, POTENT AND SELECTIVE KAPPA-OPIOID RECEPTOR ANTAGONISTS [J].
PORTOGHESE, PS ;
LIPKOWSKI, AW ;
TAKEMORI, AE .
LIFE SCIENCES, 1987, 40 (13) :1287-1292
[8]   PHARMACOLOGY OF DELTA-OPIOID RECEPTORS IN THE HAMSTER VAS-DEFERENS [J].
SHEEHAN, MJ ;
HAYES, AG ;
TYERS, MB .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 130 (1-2) :57-64
[9]  
TAKEMORI AE, 1985, ANNU REV PHARMACOL, V25, P193
[10]   A CLASSIFICATION OF OPIATE RECEPTORS THAT MEDIATE ANTINOCICEPTION IN ANIMALS [J].
TYERS, MB .
BRITISH JOURNAL OF PHARMACOLOGY, 1980, 69 (03) :503-512