EFFECT OF CERTAIN TABLET FORMULATION FACTORS ON DISSOLUTION RATE OF ACTIVE INGREDIENT .1. IMPORTANCE OF USING APPROPRIATE AGITATION INTENSITIES FOR IN VITRO DISSOLUTION RATE MEASUREMENTS TO REFLECT IN VIVO CONDITIONS

被引:137
作者
LEVY, G
机构
关键词
D O I
10.1002/jps.2600521105
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:1039 / &
相关论文
共 24 条
[1]   A PRELIMINARY REPORT OF THE EFFECT OF GASTRIC MUCOUS UPON TABLET DISINTEGRATION [J].
ABBOTT, DD ;
PACKMAN, EW ;
REES, EW ;
HARRISSON, JWE .
JOURNAL OF THE AMERICAN PHARMACEUTICAL ASSOCIATION, 1959, 48 (01) :19-21
[2]   KINETICS OF SOLUTION IN HIGH VISCOSITY LIQUIDS - SODIUM CHLORIDE-GLYCEROL [J].
COOPER, AR ;
KINGERY, WD .
JOURNAL OF PHYSICAL CHEMISTRY, 1962, 66 (04) :665-&
[3]  
DAVENPORT HW, 1961, PHYSIOLOGY DIGESTIVE, pCH3
[4]  
DAVION M, 1953, THESIS U PARIS
[5]   EFFECTS OF BUFFERED AND UNBUFFERED ACETYLSALICYLIC ACID UPON GASTRIC ACIDITY OF NORMAL HUMAN SUBJECTS [J].
DAVISON, C ;
SMITH, BW ;
SMITH, PK .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1962, 51 (08) :759-&
[6]   THE DISSOLUTION AND DIFFUSION OF ASPIRIN IN AQUEOUS MEDIA [J].
EDWARDS, LJ .
TRANSACTIONS OF THE FARADAY SOCIETY, 1951, 47 (11) :1191-1210
[7]   LOS OF SENSITIVITY IN DISTINGUISHING REAL DIFFERENCES IN DISSOLUTION RATES DUE TO INCREASING INTENSITY OF AGITATION [J].
HAMLIN, WE ;
BALLARD, BE ;
WAGNER, JG ;
NELSON, E .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1962, 51 (05) :432-&
[8]  
IVY AC, 1950, PEPTIC ULCER, P42
[9]   EFFECT OF CERTAIN TABLET FORMULATION FACTORS ON DISSOLUTION RATE OF ACTIVE INGREDIENT .2. GRANULE SIZE, STARCH CONCENTRATION, AND COMPRESSION PRESSURE [J].
LEVY, G ;
WHITE, DC ;
ANTKOWIAK, JM ;
PROCKNAL, JA .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1963, 52 (11) :1047-&
[10]   PHYSICOCHEMICAL BASIS OF THE BUFFERED ACETYLSALICYLIC ACID CONTROVERSY [J].
LEVY, G ;
HAYES, BA .
NEW ENGLAND JOURNAL OF MEDICINE, 1960, 262 (21) :1053-1058