CYCLIC AND ACYCLIC PARTIAL RETRO-INVERSO ENKEPHALINAMIDES - MU RECEPTOR SELECTIVE ENZYME RESISTANT ANALOGS

被引：32

作者：

BERMAN, JM ^{[1
]}

GOODMAN, M ^{[1
]}

NGUYEN, TMD ^{[1
]}

SCHILLER, PW ^{[1
]}

机构：

[1] CLIN RES INST MONTREAL, MONTREAL H2W 1R7, QUEBEC, CANADA

来源：

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS | 1983年 / 115卷 / 03期

关键词：

D O I：

10.1016/S0006-291X(83)80014-X

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：864 / 870

页数：7

共 19 条

[1]

BERMAN JM, UNPUB INT J PEPTIDE

[2]

CHANG KJ, 1979, J BIOL CHEM, V254, P2610

[3]

CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099

[4] SYNTHESIS AND PHARMACOLOGICAL CHARACTERIZATION INVITRO OF CYCLIC ENKEPHALIN ANALOGS - EFFECT OF CONFORMATIONAL CONSTRAINTS ON OPIATE RECEPTOR SELECTIVITY [J].

DIMAIO, J ;

NGUYEN, TMD ;

LEMIEUX, C ;

SCHILLER, PW .

JOURNAL OF MEDICINAL CHEMISTRY, 1982, 25 (12) :1432-1438

[5] A CYCLIC ENKEPHALIN ANALOG WITH HIGH INVITRO OPIATE ACTIVITY [J].

DIMAIO, J ;

SCHILLER, PW .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (12) :7162-7166

[6]

GOODMAN M, 1981, PERSPECTIVES PEPTIDE, P283

[7] MODE OF DEACTIVATION OF ENKEPHALINS BY RAT AND HUMAN-PLASMA AND RAT-BRAIN HOMOGENATES [J].

HAMBROOK, JM ;

MORGAN, BA ;

RANCE, MJ ;

SMITH, CFC .

NATURE, 1976, 262 (5571) :782-783

[8]

HANDA BK, 1981, EUR J PHARMACOL, V70, P731

[9] CONFORMATIONAL RESTRICTIONS OF BIOLOGICALLY-ACTIVE PEPTIDES VIA AMINO-ACID SIDE-CHAIN GROUPS [J].

HRUBY, VJ .

LIFE SCIENCES, 1982, 31 (03) :189-199

[10] IDENTIFICATION OF 2 RELATED PENTAPEPTIDES FROM BRAIN WITH POTENT OPIATE AGONIST ACTIVITY [J].

HUGHES, J ;

SMITH, TW ;

KOSTERLITZ, HW ;

FOTHERGILL, LA ;

MORGAN, BA ;

MORRIS, HR .

NATURE, 1975, 258 (5536) :577-579

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