ENZYME ASSISTED PREPARATION OF ENANTIOMERICALLY PURE BETA-ADRENERGIC BLOCKERS .2. BUILDING-BLOCKS OF HIGH OPTICAL PURITY AND THEIR SYNTHETIC CONVERSION

被引：41

作者：

ADER, U ^{[1
]}

SCHNEIDER, MP ^{[1
]}

机构：

[1] UNIV GESAMTHSCH WUPPERTAL,FACBERCICH BERG 9,W-5600 WUPPERTAL 1,GERMANY

来源：

TETRAHEDRON-ASYMMETRY | 1992年 / 3卷 / 02期

关键词：

D O I：

10.1016/S0957-4166(00)80191-3

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

Based on previous screening results a series of potential building blocks 2-4 for beta-adrenergic blockers were prepared both by enzymatic hydrolysis and acyltransfer and further transformed into the corresponding oxiranes and aminoalcohols of defined absolute configurations.

引用

页码：205 / 208

页数：4

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