Synthesis of new pyrazoline and pyrazole derivatives

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作者
Basaif, SA
Albar, HA
Faidallah, HM
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O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Condensation of p-sulfamylphenylhydrazine with chalcones, leads either to hydrazones (2) or pyrazolines (3). Oxidation of (3) afforded pyrazole derivatives (4). Benzenesulfonylureas (5) and thioureas (6) were also prepared, and (6) was converted to the corresponding thiazolidinones (7) on reaction with ethyl bromoacetate.
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页码:121 / 124
页数:4
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