EVALUATION OF PROTEIN-N-(2-HYDROXYPROPYL)METHACRYLAMIDE COPOLYMER CONJUGATES AS TARGETABLE DRUG CARRIERS .1. BINDING, PINOCYTIC UPTAKE AND INTRACELLULAR-DISTRIBUTION OF TRANSFERRIN AND ANTI-TRANSFERRIN RECEPTOR ANTIBODY CONJUGATES

被引:33
作者
FLANAGAN, PA
KOPECKOVA, P
KOPECEK, J
DUNCAN, R
机构
[1] UNIV KEELE, DEPT BIOL SCI, CANC RES CAMPAIGN LAB, KEELE ST5 5BG, STAFFS, ENGLAND
[2] CZECHOSLOVAK ACAD SCI, INST MACROMOLEC CHEM, CS-11142 PRAGUE 1, CZECHOSLOVAKIA
关键词
D O I
10.1016/0304-4165(89)90146-3
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:83 / 91
页数:9
相关论文
共 43 条
[1]  
CARTLIDGE S A, 1986, Journal of Controlled Release, V3, P55, DOI 10.1016/0168-3659(86)90064-7
[2]  
COURTENAYLUCK NS, 1986, CANCER RES, V46, P6489
[3]   ANTICANCER AGENTS COUPLED TO N-(2-HYDROXYPROPYL)METHACRYLAMIDE COPOLYMERS .2. EVALUATION OF DAUNOMYCIN CONJUGATES INVIVO AGAINST L1210 LEUKEMIA [J].
DUNCAN, R ;
KOPECKOVA, P ;
STROHALM, J ;
HUME, IC ;
LLOYD, JB ;
KOPECEK, J .
BRITISH JOURNAL OF CANCER, 1988, 57 (02) :147-156
[4]  
DUNCAN R, 1983, MAKROMOL CHEM, V184, P1997
[5]   FATE OF N-(2-HYDROXYPROPYL)METHACRYLAMIDE COPOLYMERS WITH PENDENT GALACTOSAMINE RESIDUES AFTER INTRAVENOUS ADMINISTRATION TO RATS [J].
DUNCAN, R ;
SEYMOUR, LCW ;
SCARLETT, L ;
LLOYD, JB ;
REJMANOVA, P ;
KOPECEK, J .
BIOCHIMICA ET BIOPHYSICA ACTA, 1986, 880 (01) :62-71
[6]   DRUG TARGETING TO LYSOSOMES [J].
DUNCAN, R ;
KOPECEK, J ;
LLOYD, JB .
BIOCHEMICAL SOCIETY TRANSACTIONS, 1984, 12 (06) :913-915
[7]   EFFECT OF MOLECULAR-SIZE OF I-125-LABELED POLY(VINYLPYRROLIDONE) ON ITS PINOCYTOSIS BY RAT VISCERAL YOLK SACS AND RAT PERITONEAL-MACROPHAGES [J].
DUNCAN, R ;
PRATTEN, MK ;
CABLE, HC ;
RINGSDORF, H ;
LLOYD, JB .
BIOCHEMICAL JOURNAL, 1981, 196 (01) :49-55
[8]  
DUNCAN R, 1986, CRIT REV BIOCOMPAT, V2, P127
[9]   DEGRADATION OF SIDE-CHAINS OF N-(2-HYDROXYPROPYL) METHACRYLAMIDE CO-POLYMERS BY LYSOSOMAL-ENZYMES [J].
DUNCAN, R ;
LLOYD, JB ;
KOPECEK, J .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1980, 94 (01) :284-290
[10]   TYROSINAMIDE RESIDUES ENHANCE PINOCYTIC CAPTURE OF N-(2-HYDROXYPROPYL)METHACRYLAMIDE COPOLYMERS [J].
DUNCAN, R ;
CABLE, HC ;
REJMANOVA, P ;
KOPECEK, J ;
LLOYD, JB .
BIOCHIMICA ET BIOPHYSICA ACTA, 1984, 799 (01) :1-8