A NEW HIGHLY POTENT PARATHYROID-HORMONE ANTAGONIST - [D-TRP12, TYR34]BPTH-(7--34)NH2

被引:65
作者
GOLDMAN, ME
MCKEE, RL
CAULFIELD, MP
REAGAN, JE
LEVY, JJ
GAY, CT
DEHAVEN, PA
ROSENBLATT, M
CHOREV, M
机构
关键词
D O I
10.1210/endo-123-5-2597
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:2597 / 2599
页数:3
相关论文
共 11 条
[1]   SOME QUANTITATIVE USES OF DRUG ANTAGONISTS [J].
ARUNLAKSHANA, O ;
SCHILD, HO .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (01) :48-58
[2]  
CHOREV M, 1988, PEPTIDE CHEM PROTEIN, P621
[3]   EVALUATION OF NOVEL PARATHYROID-HORMONE ANALOGS USING A BOVINE RENAL MEMBRANE-RECEPTOR BINDING ASSAY [J].
GOLDMAN, ME ;
CHOREV, M ;
REAGAN, JE ;
NUTT, RF ;
LEVY, JJ ;
ROSENBLATT, M .
ENDOCRINOLOGY, 1988, 123 (03) :1468-1475
[4]   INVIVO STUDIES ON AN ANTAGONIST OF PARATHYROID-HORMONE [NLE-8,NLE-18,TYR-34]BPTH-(3-34)AMIDE [J].
GRAY, DA ;
PARSONS, JA ;
POTTS, JT ;
ROSENBLATT, M ;
STEVENSON, RW .
BRITISH JOURNAL OF PHARMACOLOGY, 1982, 76 (02) :259-263
[5]  
HORUCHI N, 1983, SCIENCE, V220, P1053
[6]   THE 7-34-FRAGMENT OF HUMAN HYPERCALCEMIA FACTOR IS A PARTIAL AGONIST ANTAGONIST FOR PARATHYROID HORMONE-STIMULATED CAMP PRODUCTION [J].
MCKEE, RL ;
GOLDMAN, ME ;
CAULFIELD, MP ;
DEHAVEN, PA ;
LEVY, JJ ;
NUTT, RF ;
ROSENBLATT, M .
ENDOCRINOLOGY, 1988, 122 (06) :3008-3010
[7]   PARATHYROID-HORMONE - CHEMISTRY, BIOSYNTHESIS, AND MODE OF ACTION [J].
POTTS, JT ;
KRONENBERG, HM ;
ROSENBLATT, M .
ADVANCES IN PROTEIN CHEMISTRY, 1982, 35 :323-396
[8]   IDENTIFICATION OF A RECEPTOR-BINDING REGION IN PARATHYROID-HORMONE [J].
ROSENBLATT, M ;
SEGRE, GV ;
TYLER, GA ;
SHEPARD, GL ;
NUSSBAUM, SR ;
POTTS, JT .
ENDOCRINOLOGY, 1980, 107 (02) :545-550
[9]  
ROSENBLATT M, 1977, J BIOL CHEM, V252, P5847
[10]  
ROSENBLATT M, 1986, NEW ENGL J MED, V315, P1004