SOME DERIVATIVES OF 1,2,3-TRIAZOLES - SYNTHESIS AND STUDY OF ANTIMICROBIAL ACTIVITY

被引：0
|
作者：
KARIMKULOV, KM
DZHURAYEV, AD
MAKHSUMOV, AG
AMANOV, N
机构：
来源：
KHIMIKO-FARMATSEVTICHESKII ZHURNAL | 1991年 / 25卷 / 06期
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中图分类号：
R9 [药学];
学科分类号：
1007 ;
摘要：
1, 2, 3-Triazoles of acetylenic esters of benzoic acid derivatives were synthesized and assayed for antimicrobial activity. They were found to have some antimicrobial activity. The highest activity was exhibited by 1-phenyl-4,5-bis-(3-bromobenzoyloxymethyl)-1,2,3-triazole which was 1.5- fold potent as compared with the well-known antimicrobial agents penicillin, levomycetin (chloramphenicol), and polymyxin.
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页码：40 / 42
页数：3
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