A PARTIAL AGONIST AT THE ANTICONVULSANT BENZODIAZEPINE RECEPTOR - REVERSAL OF THE ANTICONVULSANT EFFECTS OF RO-15-1788 WITH CGS-8216

被引:31
作者
ROBERTSON, HA
RIIVES, M
BLACK, DAS
PETERSON, MR
机构
关键词
D O I
10.1016/0006-8993(84)91275-7
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:388 / 390
页数:3
相关论文
共 13 条
[1]   MODIFICATION OF THE ANTICONVULSANT EFFICACY OF DIAZEPAM BY RO-15-1788 IN THE KINDLED AMYGDALOID SEIZURE MODEL [J].
ALBERTSON, TE ;
BOWYER, JF ;
PAULE, MG .
LIFE SCIENCES, 1982, 31 (15) :1597-1601
[2]   INTERACTION OF CONVULSIVE LIGANDS WITH BENZODIAZEPINE RECEPTORS [J].
BRAESTRUP, C ;
SCHMIECHEN, R ;
NEEF, G ;
NIELSEN, M ;
PETERSEN, EN .
SCIENCE, 1982, 216 (4551) :1241-1243
[3]   CGS-8216 - RECEPTOR-BINDING CHARACTERISTICS OF A POTENT BENZODIAZEPINE ANTAGONIST [J].
CZERNIK, AJ ;
PETRACK, B ;
KALINSKY, HJ ;
PSYCHOYOS, S ;
CASH, WD ;
TSAI, C ;
RINEHART, RK ;
GRANAT, FR ;
LOVELL, RA ;
BRUNDISH, DE ;
WADE, R .
LIFE SCIENCES, 1982, 30 (04) :363-372
[4]   ANXIOGENIC AND NON-ANXIOGENIC BENZODIAZEPINE ANTAGONISTS [J].
DECARVALHO, LP ;
GRECKSCH, G ;
CHAPOUTHIER, G ;
ROSSIER, J .
NATURE, 1983, 301 (5895) :64-66
[5]   PROCONVULSANT ACTION OF CGS 8216 [J].
FILE, SE .
NEUROSCIENCE LETTERS, 1983, 35 (03) :317-320
[6]   PK 8165 AND PK 9084, 2 QUINOLINE DERIVATIVES WITH ANXIOLYTIC PROPERTIES, ANTAGONIZE THE ANTI-CONVULSANT EFFECTS OF DIAZEPAM [J].
GEE, KW ;
BRINTON, RE ;
YAMAMURA, HI .
BRAIN RESEARCH, 1983, 264 (01) :168-172
[7]  
GREKSCH G, 1983, LIFE SCI, V32, P2579
[8]   SELECTIVE ANTAGONISTS OF BENZODIAZEPINES [J].
HUNKELER, W ;
MOHLER, H ;
PIERI, L ;
POLC, P ;
BONETTI, EP ;
CUMIN, R ;
SCHAFFNER, R ;
HAEFELY, W .
NATURE, 1981, 290 (5806) :514-516
[9]   MULTIPLE BENZODIAZEPINE RECEPTORS - EVIDENCE OF A DISSOCIATION BETWEEN ANTI-CONFLICT AND ANTICONVULSANT PROPERTIES BY PK8165 AND PK9084 (2 QUINOLINE DERIVATIVES) [J].
LEFUR, G ;
MIZOULE, J ;
BURGEVIN, MC ;
FERRIS, O ;
HEAULME, M ;
GAUTHIER, A ;
GUEREMY, C ;
UZAN, A .
LIFE SCIENCES, 1981, 28 (13) :1439-1448
[10]   AGONIST AND ANTAGONIST BENZODIAZEPINE RECEPTOR INTERACTION INVITRO [J].
MOHLER, H ;
RICHARDS, JG .
NATURE, 1981, 294 (5843) :763-765