[I-125]-1-(2,5-DIMETHOXY-4-IODOPHENYL)-2-AMINOPROPANE - AN IODINATED RADIOLIGAND THAT SPECIFICALLY LABELS THE AGONIST HIGH-AFFINITY STATE OF 5-HT2 SEROTONIN RECEPTORS

被引：116

作者：

GLENNON, RA ^{[1
]}

SEGGEL, MR ^{[1
]}

SOINE, WH ^{[1
]}

HERRICKDAVIS, K ^{[1
]}

LYON, RA ^{[1
]}

TITELER, M ^{[1
]}

机构：

[1] UNION UNIV ALBANY MED COLL,DEPT PHARMACOL & TOXICOL,ALBANY,NY 12208

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1988年 / 31卷 / 01期

关键词：

D O I：

10.1021/jm00396a003

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：5 / 7

页数：3

共 10 条

[1]

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[2] BEHAVIORAL AND SEROTONIN RECEPTOR PROPERTIES OF 4-SUBSTITUTED DERIVATIVES OF THE HALLUCINOGEN 1-(2,5-DIMETHOXYPHENYL)-2-AMINOPROPANE [J].

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[5] PREPARATION AND PURIFICATION OF 7-IODOCLONAZEPAM FOR USE IN RADIOIMMUNOASSAY [J].

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[7]

LYON RA, 1987, MOL PHARMACOL, V31, P194

[8]

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[9] SELECTIVITY OF SEROTONERGIC DRUGS FOR MULTIPLE BRAIN-SEROTONIN RECEPTORS - ROLE OF [H-3] 4-BROMO-2,5-DIMETHOXYPHENYLISOPROPYLAMINE ([H-3]DOB), A 5-HT2 AGONIST RADIOLIGAND [J].

TITELER, M ;

LYON, RA ;

DAVIS, KH ;

GLENNON, RA .

BIOCHEMICAL PHARMACOLOGY, 1987, 36 (19) :3265-3271

[10] [H-3]DOB - A SPECIFIC AGONIST RADIOLIGAND FOR 5-HT2 SEROTONIN RECEPTORS [J].

TITELER, M ;

HERRICK, K ;

LYON, RA ;

MCKENNEY, JD ;

GLENNON, RA .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 117 (01) :145-146

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