HIV PROTEINASE-INHIBITORS

被引:24
作者
ROBERTS, NA
CRAIG, JC
DUNCAN, IB
机构
关键词
D O I
10.1042/bst0200513
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:513 / 516
页数:4
相关论文
共 26 条
[1]  
BILLICH S, 1988, J BIOL CHEM, V263, P17905
[2]  
CRAIG J C, 1991, Antiviral Chemistry and Chemotherapy, V2, P181
[3]   ANTIVIRAL PROPERTIES OF RO 31-8959, AN INHIBITOR OF HUMAN-IMMUNODEFICIENCY-VIRUS (HIV) PROTEINASE [J].
CRAIG, JC ;
DUNCAN, IB ;
HOCKLEY, D ;
GRIEF, C ;
ROBERTS, NA ;
MILLS, JS .
ANTIVIRAL RESEARCH, 1991, 16 (04) :295-305
[4]   INHIBITION OF HUMAN IMMUNODEFICIENCY VIRUS-1 PROTEASE INVITRO - RATIONAL DESIGN OF SUBSTRATE-ANALOG INHIBITORS [J].
DREYER, GB ;
METCALF, BW ;
TOMASZEK, TA ;
CARR, TJ ;
CHANDLER, AC ;
HYLAND, L ;
FAKHOURY, SA ;
MAGAARD, VW ;
MOORE, ML ;
STRICKLER, JE ;
DEBOUCK, C ;
MEEK, TD .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1989, 86 (24) :9752-9756
[5]   SELECTIVE PHOSPHINATE TRANSITION-STATE ANALOG INHIBITORS OF THE PROTEASE OF HUMAN-IMMUNODEFICIENCY-VIRUS [J].
GROBELNY, D ;
WONDRAK, EM ;
GALARDY, RE ;
OROSZLAN, S .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1990, 169 (03) :1111-1116
[6]   ELECTRON-MICROSCOPY OF HUMAN IMMUNODEFICIENCY VIRUS [J].
HOCKLEY, DJ ;
WOOD, RD ;
JACOBS, JP ;
GARRETT, AJ .
JOURNAL OF GENERAL VIROLOGY, 1988, 69 :2455-2469
[7]  
HOLMES H C, 1991, Antiviral Chemistry and Chemotherapy, V2, P287
[8]   MURINE LEUKEMIA-VIRUS MATURATION - PROTEASE REGION REQUIRED FOR CONVERSION FROM IMMATURE TO MATURE CORE FORM AND FOR VIRUS INFECTIVITY [J].
KATOH, I ;
YOSHINAKA, Y ;
REIN, A ;
SHIBUYA, M ;
ODAKA, T ;
OROSZLAN, S .
VIROLOGY, 1985, 145 (02) :280-292
[9]  
KEMPF DJ, 1990, J MED CHEM, V33, P2657
[10]   ACTIVE HUMAN IMMUNODEFICIENCY VIRUS PROTEASE IS REQUIRED FOR VIRAL INFECTIVITY [J].
KOHL, NE ;
EMINI, EA ;
SCHLEIF, WA ;
DAVIS, LJ ;
HEIMBACH, JC ;
DIXON, RAF ;
SCOLNICK, EM ;
SIGAL, IS .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1988, 85 (13) :4686-4690