COMPETITION BETWEEN LIDOCAINE AND ONE OF ITS METABOLITES, GLYCYLXYLIDIDE, FOR CARDIAC SODIUM-CHANNELS

被引:26
作者
BENNETT, PB [1 ]
WOOSLEY, RL [1 ]
HONDEGHEM, LM [1 ]
机构
[1] VANDERBILT UNIV,MED CTR,SCH MED,DEPT MED,NASHVILLE,TN 37232
关键词
D O I
10.1161/01.CIR.78.3.692
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:692 / 700
页数:9
相关论文
共 24 条
[1]   LIDOCAINE BLOCK OF CARDIAC SODIUM-CHANNELS [J].
BEAN, BP ;
COHEN, CJ ;
TSIEN, RW .
JOURNAL OF GENERAL PHYSIOLOGY, 1983, 81 (05) :613-642
[2]  
Bevington P.R., 1969, DATA REDUCTION ERROR
[3]   LIPID SOLUBILITY MODULATES PH POTENTIATION OF LOCAL-ANESTHETIC BLOCK OF VMAX REACTIVATION IN GUINEA-PIG MYOCARDIUM [J].
BROUGHTON, A ;
GRANT, AO ;
STARMER, CF ;
KLINGER, JK ;
STAMBLER, BS ;
STRAUSS, HC .
CIRCULATION RESEARCH, 1984, 55 (04) :513-523
[4]  
BROWN AM, 1981, J PHYSIOL-LONDON, V318, P479
[5]  
BROWN AM, 1981, J PHYSIOL-LONDON, V318, P455
[6]   INTERACTIONS BETWEEN QUATERNARY LIDOCAINE, THE SODIUM-CHANNEL GATES, AND TETRODOTOXIN [J].
CAHALAN, MD ;
ALMERS, W .
BIOPHYSICAL JOURNAL, 1979, 27 (01) :39-55
[7]   LIGNOCAINE THERAPY FOR VENTRICULAR ECTOPIC ACTIVITY AFTER ACUTE MYOCARDIAL INFARACTION - DOUBLE-BLIND TRIAL [J].
CHOPRA, MP ;
THADANI, U ;
PORTAL, RW ;
ABER, CP .
BRITISH MEDICAL JOURNAL, 1971, 3 (5776) :668-&
[8]   LIGNOCAINE THERAPY AFTER ACUTE MYOCARDIAL INFARCTION [J].
CHOPRA, MP ;
PORTAL, RW ;
ABER, CP .
BRITISH MEDICAL JOURNAL, 1969, 1 (5638) :213-&
[9]   EVIDENCE FOR A SPECIFIC RECEPTOR-SITE FOR LIDOCAINE, QUINIDINE, AND BUPIVACAINE ASSOCIATED WITH CARDIAC SODIUM-CHANNELS IN GUINEA-PIG VENTRICULAR MYOCARDIUM [J].
CLARKSON, CW ;
HONDEGHEM, LM .
CIRCULATION RESEARCH, 1985, 56 (04) :496-506
[10]   ISOLATION OF CALCIUM TOLERANT MYOCYTES FROM ADULT-RAT HEARTS - REVIEW OF THE LITERATURE AND DESCRIPTION OF A METHOD [J].
FARMER, BB ;
MANCINA, M ;
WILLIAMS, ES ;
WATANABE, AM .
LIFE SCIENCES, 1983, 33 (01) :1-18